Activation of Toll-like receptor 9 and production of epitope specific antibody by liposome-encapsulated CpG-DNA

BMB Rep. 2011 Sep;44(9):607-12. doi: 10.5483/bmbrep.2011.44.9.607.

Abstract

Several investigators have shown that CpG-DNA has outstanding effects as a Th1-responsive adjuvant and that its potent adjuvant effects are enhanced by encapsulation with a liposome of proper composition. In this study, we showed that encapsulation with phosphatidyl-Β-oleoyl-γ-palmitoyl ethanolamine (DOPE): cholesterol hemisuccinate (CHEMS) complex enhances the immunostimulatory activity of CpG DNA and the binding of CpG-DNA to TLR9. We also examined involvement of myeloid differentiation protein (MyD88) and NF-κB activation in liposome-encapsulated CpG-DNA-induced IL-8 promoter activation. In this manuscript, the natural phosphodiester bond CpG-DNA encapsulated by DOPE : CHEMS complex is designated as Lipoplex(O). Importantly, we successfully screened B cell epitopes of envelope protein (E protein) of hepatitis C virus (HCV-E) and attachment glycoprotein G of human respiratory syncytial virus (HRSV-G) by immunization with complexes of several peptides and Lipoplex(O) without carriers. Therefore, Lipoplex(O) is potentially applicable as a universal adjuvant for peptide-based epitope screening and antibody production.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adjuvants, Immunologic
  • Antibodies / immunology
  • Antibodies / metabolism*
  • Cholesterol Esters / chemistry
  • CpG Islands / immunology*
  • DNA / immunology*
  • DNA / metabolism
  • Epitopes / immunology*
  • Hepacivirus / metabolism
  • Humans
  • Interleukin-8 / genetics
  • Interleukin-8 / metabolism
  • Liposomes / chemistry*
  • Myeloid Differentiation Factor 88 / metabolism
  • NF-kappa B / metabolism
  • Peptides / immunology
  • Peptides / metabolism
  • Phosphatidylethanolamines / chemistry
  • Promoter Regions, Genetic
  • Protein Binding
  • Toll-Like Receptor 9 / metabolism*
  • Viral Envelope Proteins / immunology
  • Viral Envelope Proteins / metabolism

Substances

  • 1,2-dioleoyl-glycero-3-phosphatidyl ethanolamine
  • Adjuvants, Immunologic
  • Antibodies
  • Cholesterol Esters
  • Epitopes
  • Interleukin-8
  • Liposomes
  • Myeloid Differentiation Factor 88
  • NF-kappa B
  • Peptides
  • Phosphatidylethanolamines
  • Toll-Like Receptor 9
  • Viral Envelope Proteins
  • DNA
  • cholesteryl succinate