Vitamin D receptor interaction with specific DNA requires a nuclear protein and 1,25-dihydroxyvitamin D3

Proc Natl Acad Sci U S A. 1990 Dec;87(24):9751-5. doi: 10.1073/pnas.87.24.9751.

Abstract

The regulation of osteocalcin gene expression by 1,25-dihydroxyvitamin D3 is mediated by the vitamin D receptor and a cis-acting DNA response element that has been identified within the 5' region of the osteocalcin promoter. In this report, we show that vitamin D receptors derived from nuclear extracts of mammalian cells bind directly to this cis-acting element in vitro and do so in a manner requiring hormone. Vitamin D receptors derived from reticulocyte lysate translations in vitro or from extracts of a Saccharomyces cerevisiae strain that expresses the recombinant protein also bind the osteocalcin responsive element, but only when nuclear extracts of mammalian cells are provided. The vitamin-D-receptor-DNA-binding accessory factor is isolated by salt extraction, labile to temperature, and sensitive to tryptic digestion. These studies suggest that the high-affinity interaction of the vitamin D receptor with the osteocalcin vitamin D response element in vitro requires both 1,25-dihydroxyvitamin D3 and an accessory protein derived from the mammalian cell nucleus.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Base Sequence
  • Calcitriol / pharmacology*
  • Cell Line
  • Cell Nucleus / metabolism
  • DNA / genetics*
  • DNA / metabolism
  • Gene Expression / drug effects*
  • Molecular Sequence Data
  • Nuclear Proteins / metabolism*
  • Oligonucleotide Probes
  • Osteocalcin / genetics*
  • Plasmids
  • Promoter Regions, Genetic
  • Protein Biosynthesis
  • Receptors, Calcitriol
  • Receptors, Steroid / genetics
  • Receptors, Steroid / metabolism*
  • Transcription, Genetic
  • Transfection

Substances

  • Nuclear Proteins
  • Oligonucleotide Probes
  • Receptors, Calcitriol
  • Receptors, Steroid
  • Osteocalcin
  • DNA
  • Calcitriol