Regulation of Notch1 signaling by Delta-like ligand 1 intracellular domain through physical interaction

Mol Cells. 2011 Aug;32(2):161-5. doi: 10.1007/s10059-011-1046-y. Epub 2011 Jun 1.

Abstract

Notch signaling involves the proteolytic cleavage of the transmembrane Notch receptor after binding to its transmembrane ligands. The Delta-like ligand 1 also undergoes proteolytic cleavage upon Notch binding, resulting in the production of a free intracellular domain. In this study, we have demonstrated that the Delta-like 1 intracellular domain (Dll1-IC) specifically binds to Notch1-IC in the nucleus, thereby disrupting the association of the Notch1-IC-RBP-Jk-MAM transcription activator complex. Additionally, the Notch1-mediated blockage of the induction of MyoD is abolished by the co-expression of Dll1-IC. Collectively, our results show that Dll1-IC functions as a negative regulator in Notch signaling via the disruption of the Notch1-IC-RBP-Jk complex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium-Binding Proteins
  • Cell Differentiation / genetics
  • HEK293 Cells
  • Humans
  • Intercellular Signaling Peptides and Proteins / metabolism*
  • Membrane Proteins / metabolism*
  • Mice
  • MyoD Protein / genetics
  • MyoD Protein / metabolism*
  • Protein Binding / genetics
  • Protein Engineering
  • Protein Structure, Tertiary / genetics
  • Receptor, Notch1 / genetics
  • Receptor, Notch1 / metabolism*
  • Sequence Deletion / genetics
  • Signal Transduction / genetics
  • Transcriptional Activation
  • Transgenes / genetics

Substances

  • Calcium-Binding Proteins
  • DLK1 protein, human
  • Intercellular Signaling Peptides and Proteins
  • Membrane Proteins
  • MyoD Protein
  • Receptor, Notch1