Cytotoxic effect of TNF-alpha and abnormal regulation of cAMP in the retinoid resistant cell line U937/GTB

Anticancer Res. 1990 Mar-Apr;10(2A):433-6.

Abstract

We have studied the effect of retinoids, forskolin and TNF-alpha on two sublines of U937 cells, U937/clone 4 and U937/GTB. Retinoids induced differentiation of U937/clone 4, while the U937/GTB cells were resistant to induction of differentiation by retinoids. Retinoids effectively reduced the proliferation of both U937/clone 4 and U937/GTB, and decreased the steady state levels of c-myc mRNA in both sublines. Furthermore, the retinoid resistant U937/GTB cells were hypersensitive to the cytotoxic effect of TNF-alpha. Forskolin increased the cAMP level in the U937/clone 4 cells 14 times above basal level, but did not change the cAMP concentration in the U937/GTB cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Differentiation / drug effects
  • Cell Division / drug effects
  • Cell Line
  • Colforsin / pharmacology
  • Cyclic AMP / biosynthesis*
  • Drug Resistance
  • Leukemia, Myeloid / metabolism
  • Leukemia, Myeloid / pathology*
  • Oncogenes
  • RNA, Messenger / metabolism
  • Tretinoin / pharmacology
  • Tumor Necrosis Factor-alpha / pharmacology*
  • Vitamin A / pharmacology

Substances

  • RNA, Messenger
  • Tumor Necrosis Factor-alpha
  • Vitamin A
  • Colforsin
  • Tretinoin
  • Cyclic AMP