A role of both NF-κB pathways in expression and transcription regulation of BAFF-R gene in multiple myeloma cells

Mol Cell Biochem. 2011 Nov;357(1-2):21-30. doi: 10.1007/s11010-011-0871-9. Epub 2011 May 24.

Abstract

B-lymphocyte stimulator (BAFF) is a recently recognized member of the tumor necrosis factor ligand family (TNF) and a potent cell-survival factor expressed in many hematopoietic cells. BAFF regulates B-cell survival, differentiation, and proliferation by binding to three TNF receptors: TACI, BCMA, and BAFF-R. The mechanism involved in BAFF-R gene expression and regulation remains elusive. In this study, we examined BAFF-R gene expression, function, and regulation in multiple myeloma (KM3) cells. It was found that BAFF-BAFF-R induced cell survival by activating NF-κB1 pathway and NF-κB2 pathway. It was also found that NF-κB was an important transcription factor involved in regulating BAFF-R expression through one NF-κB binding site in the BAFF-R promoter, suggesting that inhibiting NF-κB could decrease the expression of BAFF-R mRNA and protein, and promote activity of BAFF-R gene. Our findings indicate that both NF-κB pathways are involved in the regulation of BAFF-R gene and the NF-κB-binding site of BAFF-R may be a new therapeutic target in this disease.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis
  • B-Cell Activating Factor / genetics
  • B-Cell Activating Factor / metabolism
  • B-Cell Activation Factor Receptor / genetics*
  • B-Cell Activation Factor Receptor / metabolism
  • Binding Sites
  • Cell Line, Tumor
  • Cell Survival
  • Gene Expression Regulation, Neoplastic*
  • Humans
  • Molecular Targeted Therapy
  • Multiple Myeloma / genetics*
  • NF-kappa B / genetics
  • NF-kappa B / metabolism*
  • NF-kappa B p52 Subunit / genetics
  • NF-kappa B p52 Subunit / metabolism
  • Nitriles / pharmacology
  • Promoter Regions, Genetic / genetics
  • Signal Transduction
  • Sulfones / pharmacology
  • Transcription Factor RelA / genetics
  • Transcription Factor RelA / metabolism
  • Transcription, Genetic*

Substances

  • 3-(4-methylphenylsulfonyl)-2-propenenitrile
  • B-Cell Activating Factor
  • B-Cell Activation Factor Receptor
  • NF-kappa B
  • NF-kappa B p52 Subunit
  • Nitriles
  • Sulfones
  • TNFRSF13C protein, human
  • TNFSF13B protein, human
  • Transcription Factor RelA