S-ketamine modulates hyperalgesia in patients with chronic pancreatitis pain

Reg Anesth Pain Med. 2011 May-Jun;36(3):303-7. doi: 10.1097/AAP.0b013e3182177022.

Abstract

Background and objectives: Upper abdominal pain is a dominant feature of chronic pancreatitis. A key phenomenon in this context is hyperalgesia, typically associated with N-methyl-d-aspartate receptor activation. This exploratory study evaluates acute effects of S-ketamine, a noncompetitive N-methyl-d-aspartate antagonist, in modulating generalized hyperalgesia in chronic pancreatitis pain.

Methods: In a blinded crossover trial, 10 chronic pancreatitis pain patients received S-ketamine for 3 hrs at 2 μg · kg · min or placebo infusion at an equivalent rate in randomized order. Clinical pain was assessed via visual analog scale (VAS) and short Dutch Language Version McGill Pain Questionnaire (sf-MPQ-DLV). Pressure pain thresholds (PPTs) were measured in dermatome C5, T4, dorsal T10, L1, and L4, and the sum of PPTs (SOPPT) calculated before, at end of, and after infusion.

Results: Nine patients completed the study. Median pain VAS before infusion was 29 mm at rest, 32 mm during activity; sf-MPQ-DLV score was 4. For the S-ketamine session median SOPPT change at infusion end was significantly higher than in the placebo session (218; interquartile range [IQR], 116-527, versus -123 [IQR, -330 to 24]; P = 0.005) and significant versus preinfusion values (2109 [IQR, 964-3035] vs 1914 [IQR, 842-2884]; P = 0.03). The SOPPT was unchanged versus preinfusion values and similar between groups at 1 hr after infusion end. No significant changes in VAS and sf-MPQ-DLV occurred.

Conclusions: S-ketamine infusion is more effective than placebo in increasing PPTs in chronic pancreatitis pain patients immediately after infusion. This effect did not outlast the infusion. Further research is warranted into S-ketamine use for reducing generalized hyperalgesia and chronic pancreatitis pain.

Publication types

  • Comparative Study
  • Randomized Controlled Trial

MeSH terms

  • Cross-Over Studies
  • Female
  • Humans
  • Hyperalgesia / complications
  • Hyperalgesia / drug therapy*
  • Infusions, Intravenous
  • Ketamine / administration & dosage*
  • Ketamine / chemistry
  • Male
  • Middle Aged
  • Pain / complications
  • Pain / drug therapy*
  • Pain Measurement / drug effects
  • Pain Measurement / methods
  • Pancreatitis, Chronic / complications
  • Pancreatitis, Chronic / drug therapy*
  • Receptors, N-Methyl-D-Aspartate / antagonists & inhibitors
  • Stereoisomerism

Substances

  • Receptors, N-Methyl-D-Aspartate
  • Ketamine