Conjugated polyelectrolyte-cisplatin complex nanoparticles for simultaneous in vivo imaging and drug tracking

Nanoscale. 2011 May;3(5):1997-2002. doi: 10.1039/c0nr00950d. Epub 2011 Mar 25.

Abstract

A molecular brush based on conjugated polyelectrolyte (CPE) grafted with dense poly(ethylene glycol) (PEG) chains was successfully complexed with an anticancer agent, cisplatin, to form cisplatin-loaded nanoparticles (CPE-PEG-Pt). The obtained nanoparticles have high far-red/near-infrared fluorescence and are able to release the drug in a continuous and slow manner. These nanoparticles have not only been used to visualize HepG2 cancer cells, but also served as an in vivo fluorescent imaging probe that simultaneously tracks the in vivo drug distribution in nude mice upon intravenous administration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / chemistry
  • Carcinoma, Hepatocellular / pathology*
  • Cell Line, Tumor
  • Cisplatin / administration & dosage*
  • Cisplatin / chemistry*
  • Mice
  • Mice, Nude
  • Microscopy, Fluorescence / methods*
  • Nanocapsules / chemistry
  • Nanocapsules / therapeutic use*
  • Polyethylene Glycols / chemistry*

Substances

  • Antineoplastic Agents
  • Nanocapsules
  • Polyethylene Glycols
  • Cisplatin