Entecavir as treatment for reactivation of hepatitis B in immunosuppressed patients

World J Gastroenterol. 2010 Nov 21;16(43):5447-51. doi: 10.3748/wjg.v16.i43.5447.

Abstract

Aim: To study the efficacy and safety of entecavir (ETV) as first-line therapy for hepatitis B virus (HBV) reactivation due to immunosuppression.

Methods: Four patients that were treated with different immunosuppressive regimens for hematological malignancies, who presented with HBV reactivation were treated with ETV. Clinical outcome, biochemical and virological factors, including quantitative hepatitis B surface antigen (HBsAg) were studied.

Results: In all patients, ETV induced suppression of HBV, and rapid clinical improvement without side effects. In one patient with an alanine aminotransferase (ALT) flare, tenofovir was added after 3 mo of treatment. Until death from disease progression at 6 mo after treatment initiation, this patient did not clear HBV infection. Retrospectively, it is highly probable that the patient had been non-adherent. In the other three patients, the virological responses were associated with an expeditious decrease in quantitative HBsAg titers with negativity after 2 mo, and all three had HBsAg seroconversion. In one patient, HBV DNA reached a plateau after 3 mo, before becoming undetectable after 1 year, despite early ALT normalization and undetectable quantitative HBsAg.

Conclusion: ETV seems to be effective and safe treatment for HBV reactivation. Monitoring of quantitative HBsAg might be an additional useful tool to monitor treatment response.

MeSH terms

  • Adenine / analogs & derivatives
  • Adenine / therapeutic use
  • Aged
  • Antiviral Agents / adverse effects
  • Antiviral Agents / therapeutic use*
  • Drug Therapy, Combination
  • Female
  • Guanine / adverse effects
  • Guanine / analogs & derivatives*
  • Guanine / therapeutic use
  • Hepatitis B / blood
  • Hepatitis B / drug therapy*
  • Hepatitis B / immunology*
  • Hepatitis B Surface Antigens / blood
  • Hepatitis B virus / drug effects
  • Hepatitis B virus / physiology
  • Humans
  • Immunocompromised Host*
  • Immunosuppressive Agents / pharmacology
  • Male
  • Middle Aged
  • Organophosphonates / therapeutic use
  • Retrospective Studies
  • Tenofovir
  • Treatment Outcome

Substances

  • Antiviral Agents
  • Hepatitis B Surface Antigens
  • Immunosuppressive Agents
  • Organophosphonates
  • entecavir
  • Guanine
  • Tenofovir
  • Adenine