Single-channel analysis of the electrical response of bovine aortic endothelial cells to bradykinin stimulation: contribution of a Ca2(+)-dependent K+ channel

J Hypertens Suppl. 1990 Dec;8(7):S193-201.

Abstract

The contribution of Ca2(+)-dependent K+ [K(Ca2+)] channels to the electrical response of cultured bovine aortic endothelial cells following bradykinin stimulation was investigated using the patch-clamp method in the cell-attached configuration. Results indicate (1) that bradykinin activates a voltage-insensitive K(Ca2+) channel of 40 pS in 150 mmol/l KCl through a second messenger mechanism; (2) that the time-course of the K(Ca2+) channel activation process corresponds to the time-dependent changes in cytosolic Ca2+ triggered by bradykinin; and (3) that there is a direct correlation between the cellular hyperpolarization induced by bradykinin and the activation of the K(Ca2+) channels. It is proposed that the hyperpolarization of bovine aortic endothelial cells following bradykinin stimulation is a result of the activation of K(Ca2+) channels, and not of a modification in the gating behaviour of an inward rectifying K+ channel (lk1) that is also observed in these cells. A more negative membrane potential may, in turn, enhance the Ca2+ influx involved in the bradykinin-induced Ca2+ signalling process.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bradykinin / pharmacology*
  • Calcium / physiology*
  • Cattle
  • Endothelium, Vascular / drug effects
  • Endothelium, Vascular / physiology*
  • Membrane Potentials / physiology
  • Nitric Oxide / physiology
  • Potassium Channels / physiology*
  • Second Messenger Systems / physiology*
  • Time Factors

Substances

  • Potassium Channels
  • Nitric Oxide
  • Bradykinin
  • Calcium