Neuropilin-1 mediates divergent R-Smad signaling and the myofibroblast phenotype

J Biol Chem. 2010 Oct 8;285(41):31840-8. doi: 10.1074/jbc.M110.151696. Epub 2010 Jul 30.

Abstract

The transforming growth factor-beta (TGF-β) superfamily is one of the most diversified cell signaling pathways and regulates many physiological and pathological processes. Recently, neuropilin-1 (NRP-1) was reported to bind and activate the latent form of TGF-β1 (LAP-TGF-β1). We investigated the role of NRP-1 on Smad signaling in stromal fibroblasts upon TGF-β stimulation. Elimination of NRP-1 in stromal fibroblast cell lines increases Smad1/5 phosphorylation and downstream responses as evidenced by up-regulation of inhibitor of differentiation (Id-1). Conversely, NRP-1 loss decreases Smad2/3 phosphorylation and its responses as shown by down-regulation of α-smooth muscle actin (α-SMA) and also cells exhibit more quiescent phenotypes and growth arrest. Moreover, we also observed that NRP-1 expression is increased during the culture activation of hepatic stellate cells (HSCs), a liver resident fibroblast. Taken together, our data suggest that NRP-1 functions as a key determinant of the diverse responses downstream of TGF-β1 that are mediated by distinct Smad proteins and promotes myofibroblast phenotype.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / genetics
  • Actins / metabolism
  • Animals
  • Cell Line, Transformed
  • Fibroblasts / cytology
  • Fibroblasts / metabolism*
  • Gene Expression Regulation / physiology
  • Hepatic Stellate Cells / cytology
  • Hepatic Stellate Cells / metabolism
  • Humans
  • Liver / metabolism
  • Mice
  • Mice, Knockout
  • Myoblasts / cytology
  • Myoblasts / metabolism*
  • Neuropilin-1 / genetics
  • Neuropilin-1 / metabolism*
  • Phosphorylation / physiology
  • Signal Transduction / physiology*
  • Smad Proteins, Receptor-Regulated / genetics
  • Smad Proteins, Receptor-Regulated / metabolism*
  • Transforming Growth Factor beta1 / metabolism

Substances

  • Actins
  • Smad Proteins, Receptor-Regulated
  • Transforming Growth Factor beta1
  • Neuropilin-1