The protective effects of (4R)-hexahydro-7,7-dimethyl-6-oxo-1,2,5-dithiazocine-4-carboxylic acid (SA3443), a novel cyclic disulfide, on chemically-induced acute liver injury

Jpn J Pharmacol. 1991 Feb;55(2):275-8. doi: 10.1254/jjp.55.275.

Abstract

The effects of SA3443, a novel cyclic disulfide compound, on acute liver injuries induced by carbon tetrachloride (CCl4), D-galactosamine and DL-ethionine were studied in rats or mice. SA3443 (100-300 mg/kg, p.o.) significantly suppressed the increases of serum transaminase activity and liver triglyceride content in the CCl4 or DL-ethionine-induced model. Furthermore, SA3443 (300 mg/kg, p.o.) clearly reduced the formation of hepatic lipid peroxide in CCl4-treated rats. These results indicate that SA3443 protects the liver against acute liver injury.

MeSH terms

  • Alanine Transaminase / blood
  • Animals
  • Aspartate Aminotransferases / blood
  • Azocines / pharmacology*
  • Carbon Tetrachloride
  • Chemical and Drug Induced Liver Injury
  • Disulfides / pharmacology*
  • Ethionine
  • Galactosamine
  • Lipid Peroxides / metabolism
  • Liver Diseases / prevention & control*
  • Male
  • Rats
  • Rats, Inbred Strains
  • Triglycerides / metabolism

Substances

  • Azocines
  • Disulfides
  • Lipid Peroxides
  • Triglycerides
  • SA 3443
  • Galactosamine
  • Carbon Tetrachloride
  • Aspartate Aminotransferases
  • Alanine Transaminase
  • Ethionine