Src kinases are required for a balanced production of IL-12/IL-23 in human dendritic cells activated by Toll-like receptor agonists

PLoS One. 2010 Jul 9;5(7):e11491. doi: 10.1371/journal.pone.0011491.

Abstract

Background: Pathogen recognition by dendritic cells (DC) is crucial for the initiation of both innate and adaptive immune responses. Activation of Toll-like Receptors (TLRs) by microbial molecular patterns leads to the maturation of DC, which present the antigen and activate T cells in secondary lymphoid tissues. Cytokine production by DC is critical for shaping the adaptive immune response by regulating T helper cell differentiation. It was previously shown by our group that Src kinases play a key role in cytokines production during TLR4 activation in human DC.

Principal findings: In this work we investigated the role of Src kinases during different TLRs triggering in human monocyte-derived DC (MoDC). We found that Src family kinases are important for a balanced production of inflammatory cytokines by human MoDC upon stimulation of TLR3 and 8 with their respective agonists. Disruption of this equilibrium through pharmacological inhibition of Src kinases alters the DC maturation pattern. In particular, while expression of IL-12 and other inflammatory cytokines depend on Src kinases, the induction of IL-23 and co-stimulatory molecules do not. Accordingly, DC treated with Src inhibitors are not compromised in their ability to induce CD4 T cell proliferation and to promote the Th17 subset survival but are less efficient in inducing Th1 differentiation.

Conclusions: We suggest that the pharmacological modulation of DC maturation has the potential to shape the quality of the adaptive immune response and could be exploited for the treatment of inflammation-related diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blotting, Western
  • CD4-Positive T-Lymphocytes / metabolism
  • Cells, Cultured
  • Dendritic Cells / drug effects*
  • Dendritic Cells / metabolism*
  • Flow Cytometry
  • Humans
  • Imidazoles / pharmacology
  • Interleukin-12 / biosynthesis*
  • Interleukin-23 / biosynthesis*
  • Oligonucleotide Array Sequence Analysis
  • Polymerase Chain Reaction
  • Pyrimidines / pharmacology
  • Toll-Like Receptor 3 / agonists
  • Toll-Like Receptor 3 / metabolism
  • Toll-Like Receptor 4 / agonists
  • Toll-Like Receptor 4 / metabolism
  • Toll-Like Receptor 8 / agonists
  • Toll-Like Receptor 8 / metabolism
  • Toll-Like Receptors / agonists*
  • Toll-Like Receptors / metabolism
  • src-Family Kinases / antagonists & inhibitors
  • src-Family Kinases / metabolism*

Substances

  • AG 1879
  • Imidazoles
  • Interleukin-23
  • Pyrimidines
  • Toll-Like Receptor 3
  • Toll-Like Receptor 4
  • Toll-Like Receptor 8
  • Toll-Like Receptors
  • Interleukin-12
  • src-Family Kinases
  • resiquimod