Cardiovascular activity of milk casein-derived tripeptides and plant sterols in spontaneously hypertensive rats

J Physiol Pharmacol. 2009 Dec;60(4):11-20.

Abstract

The effect of chronic treatment with fermented milk products containing bioactive tripeptides and plant sterols on blood pressure and vascular function was investigated in spontaneously hypertensive rats (SHR). Six-weeks old male SHR (n=36) were randomized into 4 groups by body weight and blood pressure to receive either Lactobacillus helveticus fermented standard milk product (containing tripeptides Ile-Pro-Pro, Val-Pro-Pro and Leu-Pro-Pro), test product with enzymatically produced tripeptides without or with plant sterols or control product without the active constituents for 8 weeks. Systolic blood pressure (SBP) was measured weekly using the tail-cuff method. Thoracic aorta and mesenteric artery were excised for vascular response measurements. At the end, SBP values vs. control product group were: standard product group -14 mmHg (P<0.05), test product group -12 mmHg and test product +sterols group -7 mmHg. The average daily tripeptide dose was 2.8-5.2 mg/kg. Total serum cholesterol in the test product +sterols group tended to be lower than in the test product group (P=0.10) whereas serum plant sterol (campesterol, sitosterol) concentrations were higher (P<0.001). In conclusion, bioactive tripeptide-containing milk products attenuated the blood pressure development in SHR. The plant sterols did not improve this effect. Vascular responses did not markedly differ between the groups, except that endothelium-derived hyperpolarizing factor (EDHF) -related aortic relaxation was demonstrated in the test product +sterols group.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholinesterase / blood
  • Animals
  • Antihypertensive Agents / analysis
  • Antihypertensive Agents / pharmacology*
  • Arteries / drug effects
  • Arteries / physiopathology
  • Blood Pressure / drug effects
  • Caseins / metabolism*
  • Cholesterol / blood
  • Cultured Milk Products* / chemistry
  • Hypertension / prevention & control*
  • Lactobacillus helveticus / metabolism
  • Male
  • Oligopeptides / analysis
  • Oligopeptides / pharmacology*
  • Phytosterols / analysis
  • Phytosterols / blood
  • Phytosterols / pharmacology*
  • Random Allocation
  • Rats
  • Rats, Inbred SHR
  • Time Factors

Substances

  • Antihypertensive Agents
  • Caseins
  • Oligopeptides
  • Phytosterols
  • isoleucyl-prolyl-proline
  • leucyl-prolyl-proline
  • valyl-prolyl-proline
  • Cholesterol
  • Acetylcholinesterase