[Swelling property of common hydrophilic polymers and their use in push-pull osmotic-pump tablets]

Zhongguo Zhong Yao Za Zhi. 2009 Sep;34(18):2319-21.
[Article in Chinese]

Abstract

Objective: To investigate the feasibility of swelling hydrogel instead of polyethylene oxide as swelling polymer in push-layer of push-pull osmotically controlled-release tablets.

Method: The swelling patterns of tablets made of pure polymers were studied by immerging the tablets into purified water and testing their size at different time points. The push-pull osmotic-pump tablets were prepared and their release patterns in vitro were studied and compared by their similar factor (f2).

Result: Tablets with different swelling materials all showed satisfying release pattern in vitro and their release ratio at 12 h were all above 80%.

Conclusion: With its release rate and cumulative release percentage at 12 h, the mixture of HPMC K15M and CMCNa in ratio of 1:1 is the best choice instead of polyethylene oxide as swelling polymer in push-layer.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Chemistry, Pharmaceutical*
  • Drug Carriers / chemistry*
  • Osmosis
  • Polymers / chemistry*
  • Tablets
  • Water / chemistry*

Substances

  • Drug Carriers
  • Polymers
  • Tablets
  • Water