Revving the Throttle on an oncogene: CDK8 takes the driver seat

Cancer Res. 2009 Oct 15;69(20):7899-901. doi: 10.1158/0008-5472.CAN-09-1704. Epub 2009 Oct 6.

Abstract

The Wnt/beta-catenin pathway plays an important role in initiation in most, if not all, colon cancers. Prior work has provided important insights into the regulation of beta-catenin stability in the cytoplasm; however, relatively little is known about the mechanism by which beta-catenin activates gene transcription in the nucleus. Using genetic approaches, studies in human colon cancers and Drosophila have identified CDK8 as a colon cancer oncogene that regulates beta-catenin transcriptional activity. These convergent observations provide new insights into the regulation of nuclear beta-catenin activity and identify a novel therapeutic target for beta-catenin-driven malignancies.

Publication types

  • Research Support, N.I.H., Extramural
  • Review

MeSH terms

  • Animals
  • Cyclin-Dependent Kinase 8 / physiology*
  • Gene Expression Regulation / physiology*
  • Humans
  • Neoplasms / genetics*
  • Neoplasms / pathology
  • Oncogenes / physiology*
  • beta Catenin / genetics*

Substances

  • beta Catenin
  • CDK8 protein, human
  • Cyclin-Dependent Kinase 8