Modulatory role for CCK-B antagonists in Parkinson's disease

Clin Neuropharmacol. 1990 Aug;13(4):339-47. doi: 10.1097/00002826-199008000-00009.

Abstract

We examined the ability of selective CCK-A and CCK-B receptor antagonists to induce or modulate the locomotor stimulant effects of dopamine agonists in MPTP-treated squirrel monkeys. Administration of 1-100 micrograms/kg i.p. of either the selective CCK-A receptor antagonist devazepide (MK-329) or the CCK-B receptor antagonist L-365,260 alone failed to stimulate a locomotor response in parkinsonian monkeys. In contrast, treatment with L-365,260 caused a 50-60% potentiation of the locomotor stimulatory effects of L-DOPA or (+)-PHNO. No such modulatory effects were observed following pretreatment with devazepide. We suggest that CCK-B receptor antagonists may be useful adjuncts to existing dopamine replacement therapy for improved management of Parkinson's disease.

MeSH terms

  • Animals
  • Benzodiazepinones / antagonists & inhibitors
  • Benzodiazepinones / pharmacology*
  • Carbidopa / pharmacology
  • Cholecystokinin / antagonists & inhibitors
  • Cholecystokinin / pharmacology*
  • Devazepide
  • Dopamine Agents / pharmacology
  • Levodopa / pharmacology
  • MPTP Poisoning
  • Male
  • Motor Activity / drug effects
  • Oxazines / pharmacology
  • Parkinson Disease, Secondary / chemically induced
  • Parkinson Disease, Secondary / physiopathology*
  • Phenylurea Compounds*
  • Receptors, Cholecystokinin / antagonists & inhibitors*
  • Receptors, Cholecystokinin / physiology
  • Saimiri

Substances

  • Benzodiazepinones
  • Dopamine Agents
  • Oxazines
  • Phenylurea Compounds
  • Receptors, Cholecystokinin
  • naxagolide
  • L 365260
  • Levodopa
  • Cholecystokinin
  • Devazepide
  • Carbidopa