Serotonin transporter binding and genotype in the nonhuman primate brain using [C-11]DASB PET

Neuroimage. 2009 Oct 1;47(4):1230-6. doi: 10.1016/j.neuroimage.2009.05.090. Epub 2009 Jun 6.

Abstract

The length polymorphism of the serotonin (5-HT) transporter gene promoter region has been implicated in altered 5-HT function and, in turn, neuropsychiatric illnesses, such as anxiety and depression. The nonhuman primate has been used as a model to study anxiety-related mechanisms in humans based upon similarities in behavior and the presence of a similar 5-HT transporter gene polymorphism. Stressful and threatening contexts in the nonhuman primate model have revealed 5-HT transporter genotype dependent differences in regional glucose metabolism. Using the rhesus monkey, we examined the extent to which serotonin transporter genotype is associated with 5-HT transporter binding in brain regions implicated in emotion-related pathology.

Methods: Genotype data and high resolution PET scans were acquired in 29 rhesus (Macaca mulatta) monkeys. [C-11]DASB dynamic PET scans were acquired for 90 min in the anesthetized animals and images of distribution volume ratio (DVR) were created to serve as a metric of 5-HT transporter binding for group comparison based on a reference region method of analysis. Regional and voxelwise statistical analysis were performed with corrections for anatomical differences in gray matter probability, sex, age and radioligand mass.

Results: There were no significant differences when comparing l/l homozygotes with s-carriers in the regions of the brain implicated in anxiety and mood related illnesses (amygdala, striatum, thalamus, raphe nuclei, temporal and prefrontal cortex). There was a significant sex difference in 5-HT transporter binding in all regions with females having 18%-28% higher DVR than males.

Conclusions: Because these findings are consistent with similar genotype findings in humans, this further strengthens the use of the rhesus model for studying anxiety-related neuropathologies.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aniline Compounds / pharmacokinetics*
  • Animals
  • Brain / diagnostic imaging*
  • Brain / metabolism*
  • Carbon Radioisotopes / pharmacokinetics
  • Female
  • Genotype
  • Humans
  • Macaca mulatta
  • Male
  • Positron-Emission Tomography / methods*
  • Protein Binding
  • Radiopharmaceuticals / pharmacokinetics
  • Serotonin Plasma Membrane Transport Proteins / metabolism*
  • Sulfides / pharmacokinetics*
  • Tissue Distribution

Substances

  • 3-amino-4-(2-dimethylaminomethylphenylsulfanyl)benzonitrile
  • Aniline Compounds
  • Carbon Radioisotopes
  • Radiopharmaceuticals
  • Serotonin Plasma Membrane Transport Proteins
  • Sulfides