Varp is a novel Rab32/38-binding protein that regulates Tyrp1 trafficking in melanocytes

Mol Biol Cell. 2009 Jun;20(12):2900-8. doi: 10.1091/mbc.e08-12-1161. Epub 2009 Apr 29.

Abstract

Two small GTPase Rabs, Rab32 and Rab38, have recently been proposed to regulate trafficking of melanogenic enzymes to melanosomes in mammalian epidermal melanocytes; however, the exact molecular mechanism of Rab32/38-mediated transport of melanogenic enzymes has never been clarified, because no Rab32/38-specific effector has ever been identified. In this study, we screened for a Rab32/38-specific effector by a yeast two-hybrid assay using a guanosine triphosphate (GTP)-locked Rab32/38 as bait and found that VPS9-ankyrin-repeat protein (Varp)/Ankrd27, characterized previously as a guanine nucleotide exchange factor (GEF) for Rab21, functions as a specific Rab32/38-binding protein in mouse melanocyte cell line melan-a. Deletion analysis showed that the first ankyrin-repeat (ANKR1) domain functions as a GTP-dependent Rab32/38-binding domain, but that the N-terminal VPS9 domain (i.e., Rab21-GEF domain) does not. Small interfering RNA-mediated knockdown of endogenous Varp in melan-a cells caused a dramatic reduction in Tyrp1 (tyrosinase-related protein 1) signals from melanosomes but did not cause any reduction in Pmel17 signals. Furthermore, expression of the ANKR1 domain in melan-a cells also caused a dramatic reduction of Tyrp1 signals, whereas the VPS9 domain had no effect. Based on these findings, we propose that Varp functions as the Rab32/38 effector that controls trafficking of Tyrp1 in melanocytes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding Sites
  • Cell Line
  • Guanine Nucleotide Exchange Factors / chemistry
  • Guanine Nucleotide Exchange Factors / deficiency
  • Guanine Nucleotide Exchange Factors / metabolism*
  • Melanocytes / cytology
  • Melanocytes / enzymology*
  • Membrane Glycoproteins / metabolism*
  • Mice
  • Molecular Sequence Data
  • Oxidoreductases / metabolism*
  • Protein Binding
  • Protein Structure, Tertiary
  • Protein Transport
  • RNA, Small Interfering / metabolism
  • Two-Hybrid System Techniques
  • rab GTP-Binding Proteins / metabolism*

Substances

  • Guanine Nucleotide Exchange Factors
  • Membrane Glycoproteins
  • RNA, Small Interfering
  • VPS9-ankyrin-repeat protein, mouse
  • Oxidoreductases
  • Tyrp1 protein, mouse
  • Rab32 protein, mouse
  • Rab38 protein, mouse
  • rab GTP-Binding Proteins

Associated data

  • GENBANK/AB455262