One-pot synthesis of N-arylpyrazoles from arylhalides

Org Lett. 2009 May 21;11(10):2097-100. doi: 10.1021/ol900515a.

Abstract

A simple one-pot method for the synthesis of diversely functionalized pyrazoles from aryl nucleophiles, di-tert-butylazodicarboxlate, and 1,3-dicarbonyl or equivalent compounds is presented.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Catalysis
  • Combinatorial Chemistry Techniques
  • Hydrocarbons, Halogenated / chemistry*
  • Molecular Structure
  • Pyrazoles / chemical synthesis*
  • Pyrazoles / chemistry

Substances

  • Hydrocarbons, Halogenated
  • Pyrazoles