The glycine brace: a component of Rab, Rho, and Ran GTPases associated with hinge regions of guanine- and phosphate-binding loops

BMC Struct Biol. 2009 Mar 5:9:11. doi: 10.1186/1472-6807-9-11.

Abstract

Background: Ras-like GTPases function as on-off switches in intracellular signalling pathways and include the Rab, Rho/Rac, Ran, Ras, Arf, Sar and G alpha families. How these families have evolutionarily diverged from each other at the sequence level provides clues to underlying mechanisms associated with their functional specialization.

Results: Bayesian analysis of divergent patterns within a multiple alignment of Ras-like GTPase sequences identifies a structural component, termed here the glycine brace, as the feature that most distinguishes Rab, Rho/Rac, Ran and (to some degree) Ras family GTPases from other Ras-like GTPases. The glycine brace consists of four residues: An aromatic residue that forms a stabilizing CH-pi interaction with a conserved glycine at the start of the guanine-binding loop; a second aromatic residue, which is nearly always a tryptophan, that likewise forms stabilizing CH-pi and NH-pi interactions with a glycine at the start of the phosphate-binding P-loop; and two other residues (typically an aspartate and a serine or threonine) that, together with a conserved buried water molecule, form a network of interactions connecting the two aromatic residues.

Conclusion: It is proposed that the two glycine residues function as hinges and that the glycine brace influences guanine nucleotide binding and release by interacting with these hinges.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Amino Acid Sequence
  • Glycine / genetics
  • Glycine / metabolism*
  • Guanine Nucleotides / metabolism*
  • Molecular Sequence Data
  • Monomeric GTP-Binding Proteins / genetics*
  • Monomeric GTP-Binding Proteins / metabolism*
  • Protein Conformation
  • Sequence Alignment
  • rab GTP-Binding Proteins / genetics
  • rab GTP-Binding Proteins / metabolism
  • ran GTP-Binding Protein / genetics
  • ran GTP-Binding Protein / metabolism
  • rho GTP-Binding Proteins / genetics
  • rho GTP-Binding Proteins / metabolism

Substances

  • Guanine Nucleotides
  • Monomeric GTP-Binding Proteins
  • rab GTP-Binding Proteins
  • ran GTP-Binding Protein
  • rho GTP-Binding Proteins
  • Glycine