Unmetabolized folic acid and total folate concentrations in breast milk are unaffected by low-dose folate supplements

Am J Clin Nutr. 2009 Jan;89(1):216-20. doi: 10.3945/ajcn.2008.26564. Epub 2008 Dec 3.

Abstract

Background: Many lactating women in North America are exposed to high synthetic folic acid intakes because of food fortification and vitamin supplement use. Few data exist on the potential long-term effect of high folic acid intakes on milk folate concentrations, whereas no data are available on the effect of supplemental [6S]-5-methyltetrahydrofolate ([6S]-5-methylTHF).

Objective: The aim of the present study was to investigate the effect of 3 treatments (placebo, folic acid, and [6S]-5-methylTHF) on milk folate and folate-binding protein (FBP) concentrations and to determine whether unmetabolized folic acid is present in milk.

Design: In this 16-wk randomized, placebo-controlled intervention, 69 lactating women were randomly assigned to receive [6S]-5-methylTHF (416 microg/d, 906 nmol/d) or a placebo, or were assigned to receive folic acid (400 microg/d, 906 nmol/d) within 1 wk postpartum. Total milk folate, FBP, and unmetabolized folic acid concentrations were measured at 16 wk.

Results: Unmetabolized folic acid was detected in 96% of milk samples tested representing approximately 8% of total milk folate concentrations. Total milk folate, FBP, and the proportion of unmetabolized milk folic acid did not differ between treatments; however, FBP concentrations were significantly lower than those published before mandatory folic acid fortification of the food supply.

Conclusion: Maternal intake of synthetic folic acid leads to the appearance of unmetabolized folic acid in milk and, seemingly, a down-regulation of milk FBP synthesis. The impact of these changes on the bioavailability of folate in infants requires further exploration.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Biological Availability
  • Carrier Proteins / metabolism*
  • Dietary Supplements
  • Double-Blind Method
  • Female
  • Folate Receptors, GPI-Anchored
  • Folic Acid / administration & dosage*
  • Folic Acid / analysis*
  • Folic Acid / metabolism
  • Food, Fortified
  • Humans
  • Lactation / metabolism*
  • Milk, Human / chemistry*
  • Pregnancy
  • Receptors, Cell Surface / metabolism*
  • Tetrahydrofolates / administration & dosage*
  • Tetrahydrofolates / analysis*
  • Tetrahydrofolates / metabolism
  • Vitamin B Complex / administration & dosage
  • Vitamin B Complex / analysis
  • Vitamin B Complex / metabolism
  • Young Adult

Substances

  • Carrier Proteins
  • Folate Receptors, GPI-Anchored
  • Receptors, Cell Surface
  • Tetrahydrofolates
  • Vitamin B Complex
  • Folic Acid
  • 5-methyltetrahydrofolate