Arkadia represses the expression of myoblast differentiation markers through degradation of Ski and the Ski-bound Smad complex in C2C12 myoblasts

Bone. 2009 Jan;44(1):53-60. doi: 10.1016/j.bone.2008.09.013. Epub 2008 Oct 7.

Abstract

The differentiation of myoblasts is regulated by multiple extracellular and intracellular factors. Of the extracellular regulators, members of transforming growth factor-beta (TGF-beta) family play critical roles in the regulation of osteoblasts and myoblast differentiation. Little is known, however, about the regulation of Myostatin/TGF-beta signaling during myoblast differentiation. In this study, we examined the roles of Arkadia, an E3 ubiquitin ligase, in Myostatin/TGF-beta signaling and the regulation of myoblast differentiation. Knockdown of Arkadia reduced Myostatin/TGF-beta signaling and enhanced the differentiation of C2C12 myoblasts. In addition, exogenous overexpression of Arkadia enhanced Myostatin/TGF-beta signaling, preventing myoblast differentiation. In the absence of the activation of Myostatin/TGF-beta signaling, knockdown of Arkadia enhanced myoblast differentiation via upregulation of Ski protein, an intracellular enhancer of myoblast differentiation. Arkadia likely affected the differentiation of myoblasts in a Smad-independent fashion by inducing Ski degradation. Knockdown of Arkadia increased the Myostatin-induced phosphorylation of Smad2/3 in C2C12 cells. Arkadia bound Smad2/3 via Ski to induce the ubiquitination of Smad2/3. These results suggest that Arkadia targets Ski-bound, inactive phospho-Smad2/3 to regulate positively Myostatin/TGF-beta signaling. Taken together, this study indicates that Arkadia regulates myoblast differentiation through both Smad-dependent and Smad-independent pathways.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biomarkers / metabolism
  • Cell Differentiation*
  • Cell Line
  • DNA-Binding Proteins / metabolism*
  • Humans
  • Mice
  • Multiprotein Complexes / metabolism
  • Myoblasts / cytology*
  • Myoblasts / metabolism*
  • Myostatin / metabolism
  • Protein Binding
  • Protein Processing, Post-Translational*
  • Proto-Oncogene Proteins / metabolism*
  • Signal Transduction
  • Smad Proteins / metabolism*
  • Smad2 Protein / metabolism
  • Smad3 Protein / metabolism
  • Transforming Growth Factor beta / metabolism
  • Ubiquitin / metabolism*
  • Ubiquitin-Protein Ligases
  • Ubiquitination

Substances

  • Biomarkers
  • DNA-Binding Proteins
  • Multiprotein Complexes
  • Myostatin
  • Proto-Oncogene Proteins
  • Ski protein, mouse
  • Smad Proteins
  • Smad2 Protein
  • Smad2 protein, mouse
  • Smad3 Protein
  • Smad3 protein, mouse
  • Transforming Growth Factor beta
  • Ubiquitin
  • Rnf111 protein, mouse
  • Ubiquitin-Protein Ligases