Dysregulated sarcoplasmic reticulum calcium release: potential pharmacological target in cardiac disease

Pharmacol Ther. 2008 Sep;119(3):340-54. doi: 10.1016/j.pharmthera.2008.06.002. Epub 2008 Jul 12.

Abstract

In the heart, Ca(2+) released from the intracellular Ca(2+) storage site, the sarcoplasmic reticulum (SR), is the principal determinant of cardiac contractility. SR Ca(2+) release is controlled by dedicated molecular machinery, composed of the cardiac ryanodine receptor (RyR2) and a number of accessory proteins, including FKBP12.6, calsequestrin (CASQ2), triadin (TRD) and junctin (JN). Acquired and genetic defects in the components of the release channel complex result in a spectrum of abnormal Ca(2+) release phenotypes ranging from arrhythmogenic spontaneous Ca(2+) releases and Ca(2+) alternans to the uniformly diminished systolic Ca(2+) release characteristic of heart failure. In this article, we will present an overview of the structure and molecular components of the SR and Ca(2+) release machinery and its modulation by different intracellular factors, such as Ca(2+) levels inside the SR as well as phosphorylation and redox modification of RyR2s. We will also discuss the relationships between abnormal SR Ca(2+) release and various cardiac disease phenotypes, including, arrhythmias and heart failure, and consider SR Ca(2+) release as a potential therapeutic target.

Publication types

  • Review

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Heart Diseases / drug therapy
  • Heart Diseases / metabolism
  • Heart Diseases / physiopathology
  • Humans
  • Models, Biological
  • Ryanodine Receptor Calcium Release Channel / physiology*
  • Sarcoplasmic Reticulum / drug effects
  • Sarcoplasmic Reticulum / metabolism*

Substances

  • Ryanodine Receptor Calcium Release Channel
  • Calcium