Cajanus cajan Linn. (Leguminosae) prevents alcohol-induced rat liver damage and augments cytoprotective function

J Ethnopharmacol. 2008 Aug 13;118(3):440-7. doi: 10.1016/j.jep.2008.05.010. Epub 2008 May 15.

Abstract

Aim of the study: Cajanus cajan Linn. (Leguminosae) is a nontoxic edible herb, widely used in Indian folk medicine for the prevention of various liver disorders. In the present study we have demonstrated that methanol-aqueous fraction (MAF2) of Cajanus cajan leaf extract could prevent the chronically treated alcohol induced rat liver damage.

Materials and methods: Chronic doses of alcohol (3.7 g/ kg) orally administered to rats for 28 days and liver function marker enzymes such as GPT, GOT, ALP and anti-oxidant enzyme activities were determined. Effect of MAF2 at a dose of 50mg/kg body weight on alcohol treated rats was noted.

Results: Alcohol effected significant increase in liver marker enzyme activities and reduced the activities of anti-oxidant enzymes. Co-administration of MAF2 reversed the liver damage due to alcohol; it decreased the activities of liver marker enzymes and augmented antioxidant enzyme activities. We also demonstrate significant decrease of the phase II detoxifying enzyme, UDP-glucuronosyl transferase (UGT) activity along with a three- and two-fold decrease of UGT2B gene and protein expression respectively. MAF2 co-administration normalized UGT activity and revived the expression of UGT2B with a concomitant expression and nuclear translocation of Nrf2, a transcription factor that regulates the expression of many cytoprotective genes.

Conclusion: Cajanus cajan extract therefore shows a promise in therapeutic use in alcohol induced liver dysfunction.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkaline Phosphatase / metabolism
  • Animals
  • Cajanus*
  • Cytoprotection*
  • Ethanol / toxicity
  • Glucuronosyltransferase / genetics
  • Liver / drug effects*
  • Male
  • NF-E2-Related Factor 2 / metabolism
  • Oxidative Stress / drug effects
  • Plant Extracts / pharmacology*
  • Plant Leaves / chemistry
  • Rats
  • Rats, Sprague-Dawley

Substances

  • NF-E2-Related Factor 2
  • Plant Extracts
  • Ethanol
  • Glucuronosyltransferase
  • Alkaline Phosphatase