Does contractile Ca2+ control calcineurin-NFAT signaling and pathological hypertrophy in cardiac myocytes?

Sci Signal. 2008 Jun 24;1(25):pe31. doi: 10.1126/scisignal.125pe31.

Abstract

In noncontractile cells, a sustained increase in total cytoplasmic Ca(2+) concentration is typically needed to activate the intracellular protein phosphatase calcineurin, leading to dephosphorylation of the transcription factor nuclear factor of activated T cells (NFAT), its nuclear translocation, and induction of gene expression. It remains a mystery exactly how Ca(2+)-dependent signaling pathways, such as that mediated by calcineurin-NFAT, are regulated in contracting cardiac myocytes given the highly specialized manner in which Ca(2+) concentration rhythmically cycles in excitation-contraction coupling. Here, we critically review evidence that supports the hypothesis that calcineurin-NFAT signaling is regulated by contractile Ca(2+) transients in cardiac myocytes.

MeSH terms

  • Calcineurin / physiology*
  • Calcium / physiology*
  • Cardiomegaly / pathology*
  • Cardiomegaly / physiopathology
  • Heart Failure / pathology
  • Heart Failure / physiopathology
  • Humans
  • Microtubules / physiology
  • Models, Biological
  • Myocytes, Cardiac / pathology*
  • Myocytes, Cardiac / physiology*
  • NFATC Transcription Factors / physiology*
  • Receptors, Adrenergic, beta / chemistry
  • Receptors, Adrenergic, beta / physiology
  • Signal Transduction

Substances

  • NFATC Transcription Factors
  • Receptors, Adrenergic, beta
  • Calcineurin
  • Calcium