Open clinical study of eye-drops containing tetrapeptides derived from substance P and insulin-like growth factor-1 for treatment of persistent corneal epithelial defects associated with neurotrophic keratopathy

Br J Ophthalmol. 2008 Jul;92(7):896-900. doi: 10.1136/bjo.2007.130013. Epub 2008 May 29.

Abstract

Background/aims: Loss of corneal sensation results in the development of persistent corneal epithelial defects. The combination of a substance P-derived peptide (FGLM-amide) and an insulin-like growth factor-1 (IGF-1)-derived peptide (SSSR) stimulates rabbit corneal epithelial migration in vitro and rabbit corneal epithelial wound closure in vivo. The clinical efficacy of eye-drops containing FGLM-amide and SSSR for the treatment of persistent corneal epithelial defects in individuals with neurotrophic keratopathy was examined in a prospective open study.

Methods: Twenty-five consecutive patients (26 eyes) with persistent corneal epithelial defects associated with neurotrophic keratopathy were treated by administration of eye-drops containing FGLM-amide and SSSR. The course of epithelial healing was monitored by slit-lamp examination.

Results: Epithelial defects resurfaced completely in 19 of the 26 eyes (73%) within 4 weeks after treatment initiation. Complete resurfacing of epithelial defects was apparent in 18 of 22 (82%) or in one of four (25%) eyes without or with limbal stem cell deficiency, respectively. No adverse effects of treatment were observed in any subject.

Conclusion: Eye-drops containing FGLM-amide and SSSR induced the rapid resurfacing of persistent epithelial defects in stem cell-positive individuals with neurotrophic keratopathy.

Publication types

  • Clinical Trial

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Cornea / innervation
  • Corneal Diseases / drug therapy*
  • Corneal Diseases / etiology
  • Corneal Diseases / pathology
  • Corneal Diseases / physiopathology
  • Drug Combinations
  • Epithelium, Corneal / pathology
  • Female
  • Humans
  • Limbus Corneae / pathology
  • Male
  • Middle Aged
  • Oligopeptides / administration & dosage
  • Oligopeptides / therapeutic use*
  • Ophthalmic Solutions
  • Prospective Studies
  • Sensation Disorders / complications
  • Sensation Disorders / drug therapy
  • Stem Cells / pathology
  • Tears / metabolism
  • Treatment Outcome
  • Visual Acuity / drug effects
  • Wound Healing / drug effects

Substances

  • Drug Combinations
  • Oligopeptides
  • Ophthalmic Solutions
  • phenylalanyl-glycyl-leucyl-methioninamide
  • seryl-seryl-seryl-arginine