Templated synthesis of single-component polymer capsules and their application in drug delivery

Nano Lett. 2008 Jun;8(6):1741-5. doi: 10.1021/nl080877c. Epub 2008 May 20.

Abstract

We report a general and facile approach for the fabrication of a new class of monodispersed, single-component and thick-walled polymer nanocapsules via the single-step assembly of macromolecules in solid core/mesoporous shell (SC/MS) silica particle templates, followed by cross-linking of the macromolecules and removal of the SC/MS templates. The general applicability of this approach is demonstrated by the preparation of nanocapsules using various polymers, including synthetic polyelectrolytes, polypeptides, and polypeptide-drug conjugates. The potential of doxorubicin (Dox)-loaded poly(L-glutamic acid) nanocapsules in tumor therapy applications is demonstrated via in vitro degradation experiments, which show a near-linear release of the Dox in the presence of a lysosomal hydrolase, nanocapsule uptake by human colorectal tumor cells, and delivery of the anticancer drug into the tumor cells, leading to tumor cell death.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / chemistry
  • Capsules
  • Cell Line
  • Cell Survival / drug effects*
  • Colorectal Neoplasms / drug therapy
  • Colorectal Neoplasms / metabolism*
  • Colorectal Neoplasms / pathology
  • Diffusion
  • Doxorubicin / administration & dosage*
  • Doxorubicin / chemistry
  • Doxorubicin / pharmacokinetics*
  • Drug Carriers / administration & dosage
  • Drug Carriers / chemistry*
  • Humans
  • Polyglutamic Acid / chemistry*

Substances

  • Antineoplastic Agents
  • Capsules
  • Drug Carriers
  • Polyglutamic Acid
  • Doxorubicin