An acidic extracellular pH induces Src kinase-dependent loss of beta-catenin from the adherens junction

Cancer Lett. 2008 Aug 18;267(1):37-48. doi: 10.1016/j.canlet.2008.03.005.

Abstract

Little attention has been paid to the role of adherens junctions (AJs) in acidic extracellular pH (pHe)-induced cell invasion. Incubation of HepG2 cells in acidic medium (pH 6.6) induced cell dispersion from tight cell clusters, and this change was accompanied by downregulation of beta-catenin at cell junctions and a rapid activation of c-Src. Pretreatment with PP2 prevented the acidic pH-induced downregulation of beta-catenin at AJ and in the membrane fractions. The acidic pHe-induced c-Src activation increased tyrosine phosphorylation of beta-catenin and decreased the amount of beta-catenin-associated E-cadherin. The depletion of membrane-bound beta-catenin coincided with enhanced cell migration and invasion, and this acidic pHe-increased cell migration and invasion was prevented by PP2. In conclusion, this study characterizes a novel signaling pathway responsible for acidic microenvironment-promoted migration and invasive behaviors of cancer cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adherens Junctions / metabolism*
  • Adherens Junctions / physiology
  • Cadherins / metabolism
  • Cell Line, Tumor
  • Cell Movement
  • Humans
  • Hydrogen-Ion Concentration*
  • Phosphorylation
  • Signal Transduction
  • beta Catenin / metabolism*
  • src-Family Kinases / pharmacology*

Substances

  • Cadherins
  • beta Catenin
  • src-Family Kinases