Isradipine therapy in chronic stable angina pectoris--comparison with nifedipine

Eur Heart J. 1991 Jul;12(7):807-12. doi: 10.1093/eurheartj/12.7.807.

Abstract

Current available calcium antagonists, although useful in angina pectoris, are often poorly tolerated. We therefore compared isradipine, a new calcium antagonist, with nifedipine in 18 patients with angina. Patients sequentially received incremental doses of either isradipine (IS) 2.5-7.5 mg three times daily or nifedipine (NF) 10-30 mg three times daily for 6 weeks each, in a randomized double-blind crossover study. Both agents produced similar (P = 0.43) increases in maximum exercise duration (IS + 30%; NF + 34%) and an equivalent (P = 0.38) increase in time to onset of angina on exercise (IS + 53%; NF + 62%). Both IS and NF significantly reduced exercise-induced ST depression (-40% and -45%) to a similar degree (P = 0.48). NF significantly (P = 0.019) reduced angina attacks (-3.0 attacks.week-1; 26%) compared to IS (-0.4; 4%) whilst a similar but non-significant trend in favour of NF was also apparent in the consumption of sublingual glyceryl trinitrate (-0.1 tablets.week-1; 2% vs +1.3.week-1; 23%; P = 0.28). However, significantly (P less than 0.03) more patients experienced adverse events whilst taking NF than with IS (36 events in 16/18 (89%) v 18 in 9/18 (50%). Thus, IS and NF increased exercise tolerance and reduced exercise angina and ST depression equally well although NF use was associated with fewer anginal episodes and IS with fewer side effects.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial

MeSH terms

  • Activities of Daily Living
  • Adult
  • Aged
  • Angina Pectoris / drug therapy*
  • Angina Pectoris / etiology
  • Angina Pectoris / physiopathology
  • Calcium Channel Blockers / administration & dosage
  • Calcium Channel Blockers / adverse effects
  • Calcium Channel Blockers / therapeutic use*
  • Double-Blind Method
  • Drug Administration Schedule
  • Electrocardiography
  • Exercise Test
  • Hemodynamics
  • Humans
  • Isradipine
  • Middle Aged
  • Nifedipine / administration & dosage
  • Nifedipine / adverse effects
  • Nifedipine / therapeutic use*
  • Pyridines / administration & dosage
  • Pyridines / adverse effects
  • Pyridines / therapeutic use*

Substances

  • Calcium Channel Blockers
  • Pyridines
  • Nifedipine
  • Isradipine