Synergism between fluoxetine and the mGlu2/3 receptor agonist, LY379268, in an in vitro model for antidepressant drug-induced neurogenesis

Neuropharmacology. 2008 Feb;54(2):428-37. doi: 10.1016/j.neuropharm.2007.10.020. Epub 2007 Nov 7.

Abstract

We examined the interaction between the selective serotonin reuptake inhibitor, fluoxetine, and group-II metabotropic glutamate (mGlu) receptors using progenitor cells isolated from cultured cerebellar granule cells, considered as an in vitro model of antidepressant-drug induced neurogenesis. These cells expressed mGlu3 receptors negatively coupled to adenylyl cyclase. A 72-h treatment with either fluoxetine or low concentrations of mGlu2/3 receptor agonists (LY379268 or 2R,4R-APDC) enhanced cell proliferation. The action of fluoxetine was mediated by the activation of 5-HT(1A) receptors. We found a strong synergism between fluoxetine and LY379268 in enhancing cell proliferation and inhibiting cAMP formation. The increased cell proliferation induced by fluoxetine+LY379268 was abrogated by the cAMP analogue, 8-Br-cAMP, as well as by drugs that inhibit the mitogen-activated protein kinase and phosphatidyilinositol-3-kinase pathways. Interestingly, fluoxetine and LY379268 also acted synergistically in promoting neuronal differentiation when progenitor cells were incubated in the presence of serum. These data support the hypothesis that a combination between classical antidepressants and mGlu2/3 receptor agonists may be helpful in the experimental treatment of depression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acids / pharmacology*
  • Animals
  • Animals, Newborn
  • Antidepressive Agents / pharmacology*
  • Bridged Bicyclo Compounds, Heterocyclic / pharmacology*
  • Cell Differentiation / drug effects
  • Cell Proliferation / drug effects
  • Cells, Cultured
  • Cerebellum / cytology
  • Cerebellum / drug effects
  • Cyclic AMP / metabolism
  • DNA, Complementary / biosynthesis
  • DNA, Complementary / genetics
  • Drug Synergism
  • Fluoxetine / pharmacology*
  • Immunohistochemistry
  • Mitogen-Activated Protein Kinases / metabolism
  • Neurons / drug effects*
  • Phosphatidylinositol 3-Kinases / metabolism
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Metabotropic Glutamate / agonists*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Selective Serotonin Reuptake Inhibitors / pharmacology*
  • Stem Cells / drug effects

Substances

  • Amino Acids
  • Antidepressive Agents
  • Bridged Bicyclo Compounds, Heterocyclic
  • DNA, Complementary
  • LY 379268
  • Receptors, Metabotropic Glutamate
  • Serotonin Uptake Inhibitors
  • Fluoxetine
  • Cyclic AMP
  • Phosphatidylinositol 3-Kinases
  • Mitogen-Activated Protein Kinases