Prolonged exposure to reduced levels of androgen accelerates prostate cancer progression in Nkx3.1; Pten mutant mice

Cancer Res. 2007 Oct 1;67(19):9089-96. doi: 10.1158/0008-5472.CAN-07-2887.

Abstract

In this report, we have investigated the relationship between androgen levels and prostate tumorigenesis in Nkx3.1; Pten mutant mice, a genetically engineered mouse model of human prostate cancer. By experimentally manipulating serum levels of testosterone in these mice for an extended period (i.e., 7 months), we have found that prolonged exposure of Nkx3.1; Pten mutant mice to androgen levels that are 10-fold lower than normal (the "Low-T" group) resulted in a marked acceleration of prostate tumorigenesis compared with those exposed to androgen levels within the reference range (the "Normal-T" group). We found that prostate tumors from the Low-T mutant mice share a similar gene expression profile as androgen-independent prostate tumors from these mutant mice, which includes the deregulated expression of several genes that are up-regulated in human hormone-refractory prostate cancer, such as Vav3 and Runx1. We propose that exposure to reduced androgens may promote prostate tumorigenesis by selecting for molecular events that promote more aggressive, hormone-refractory tumors.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Androgens / deficiency*
  • Androgens / metabolism
  • Animals
  • Disease Progression
  • Homeodomain Proteins / genetics*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Neoplasms, Hormone-Dependent / genetics*
  • Neoplasms, Hormone-Dependent / metabolism
  • Neoplasms, Hormone-Dependent / pathology
  • Orchiectomy
  • PTEN Phosphohydrolase / genetics*
  • Prostatic Neoplasms / genetics*
  • Prostatic Neoplasms / metabolism
  • Prostatic Neoplasms / pathology
  • Testosterone Propionate / pharmacology
  • Transcription Factors / genetics*

Substances

  • Androgens
  • Homeodomain Proteins
  • Nkx3-1 protein, mouse
  • Transcription Factors
  • PTEN Phosphohydrolase
  • Testosterone Propionate