Structural insight into the interaction between platelet integrin alphaIIbbeta3 and cytoskeletal protein skelemin

J Biol Chem. 2007 Nov 2;282(44):32349-56. doi: 10.1074/jbc.M704666200. Epub 2007 Sep 5.

Abstract

Skelemin is a large cytoskeletal protein critical for cell morphology. Previous studies have suggested that its two-tandem immunoglobulin C2-like repeats (SkIgC4 and SkIgC5) are involved in binding to integrin beta3 cytoplasmic tail (CT), providing a mechanism for skelemin to regulate integrin-mediated signaling and cell spreading. Using NMR spectroscopy, we have studied the molecular details of the skelemin IgC45 interaction with the cytoplasmic face of integrin alphaIIbbeta3. Here, we show that skelemin IgC45 domains form a complex not only with integrin beta3 CT but also, surprisingly, with the integrin alphaIIb CT. Chemical shift mapping experiments demonstrate that both membrane-proximal regions of alphaIIb and beta3 CTs are involved in binding to skelemin. NMR structural determinations, combined with homology modeling, revealed that SkIgC4 and SkIgC5 both exhibited a conserved Ig-fold and both repeats were required for effective binding to and attenuation of alphaIIbbeta3 cytoplasmic complex. These data provide the first molecular insight into how skelemin may interact with integrins and regulate integrin-mediated signaling and cell spreading.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Connectin
  • Integrin beta3 / metabolism*
  • Models, Molecular
  • Molecular Sequence Data
  • Muscle Proteins / chemistry*
  • Muscle Proteins / metabolism*
  • Nuclear Magnetic Resonance, Biomolecular
  • Platelet Membrane Glycoprotein IIb / metabolism*

Substances

  • Connectin
  • Integrin beta3
  • Muscle Proteins
  • Platelet Membrane Glycoprotein IIb

Associated data

  • PDB/2JTD