Highly stereoselective epoxidation of alpha-methyl-gamma-hydroxy-alpha,beta-unsaturated esters: rationalization and synthetic applications

J Org Chem. 2007 Aug 17;72(17):6614-7. doi: 10.1021/jo0709955. Epub 2007 Jul 26.

Abstract

The diastereoselectivity of the nucleophilic epoxidation of gamma-hydroxy-alpha,beta-unsaturated esters having a methyl substituent at the alpha- or beta-position was investigated. Epoxidation of the alpha-methyl-substituted enoate was highly stereoselective, giving rise to the syn isomer. This finding was used to perform an enantioselective synthesis of a natural product having a beta-hydroxy-alpha-methylene-gamma-butyrolactone motif. The nucleophilic epoxidation of enoates was found to be irreversible. Models to explain the observed stereoselectivities are proposed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Epoxy Compounds / chemistry*
  • Esters / chemistry*
  • Magnetic Resonance Spectroscopy
  • Spectrophotometry, Infrared
  • Stereoisomerism

Substances

  • Epoxy Compounds
  • Esters