3-Aminorhodanine and 2-hydrazino-2-imidazo-line hydrazones. Synthesis and antiparasitic pharmacology

Boll Chim Farm. 1991 Apr;130(4):124-7.

Abstract

Two series of hydrazones were prepared by condensation of various aldehydes with 2-aminorhodanine (series 1) and 2-hydrazino-2-imidazoline (series 2). These compounds showed interesting antiparasitic activities against amoeba, trichomonas, leishmania and plasmodium.

MeSH terms

  • Animals
  • Antiprotozoal Agents / chemical synthesis*
  • Antiprotozoal Agents / pharmacology
  • Eukaryota / drug effects
  • Hydrazones / chemical synthesis
  • Hydrazones / pharmacology
  • Imidazoles / chemical synthesis
  • Imidazoles / pharmacology
  • In Vitro Techniques
  • Microbial Sensitivity Tests
  • Rabbits
  • Rhodanine / analogs & derivatives*
  • Rhodanine / chemical synthesis
  • Rhodanine / pharmacology

Substances

  • Antiprotozoal Agents
  • Hydrazones
  • Imidazoles
  • 3-aminorhodanine
  • Rhodanine