GNL3L inhibits activity of estrogen-related receptor gamma by competing for coactivator binding

J Cell Sci. 2007 Aug 1;120(Pt 15):2532-43. doi: 10.1242/jcs.009878. Epub 2007 Jul 10.

Abstract

Guanine nucleotide binding protein-like 3 (GNL3L) is the closest homologue of a stem cell-enriched factor nucleostemin in vertebrates. They share the same yeast orthologue, Grn1p, but only GNL3L can rescue the growth-deficient phenotype in Grn1-null yeasts. To determine the unique function of GNL3L, we identified estrogen-related receptor gamma (ERRgamma) as a GNL3L-specific binding protein. GNL3L and ERRgamma are coexpressed in the eye, kidney and muscle, and co-reside in the nucleoplasm. The interaction between GNL3L and ERRgamma requires the intermediate domain of GNL3L and the AF2-domain of ERRgamma. Gain-of- and loss-of-function experiments show that GNL3L can inhibit the transcriptional activities of ERR genes in a cell-based reporter system, which does not require the nucleolar localization of GNL3L. We further demonstrate that GNL3L is able to reduce the steroid receptor coactivator (SRC) binding and the SRC-mediated transcriptional coactivation of ERRgamma. This work reveals a novel mechanism that negatively regulates the transcriptional function of ERRgamma by GNL3L through coactivator competition.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Binding, Competitive
  • Cell Nucleolus / metabolism
  • GTP-Binding Proteins / chemistry
  • GTP-Binding Proteins / metabolism*
  • Gene Expression Regulation
  • Histone Acetyltransferases / metabolism
  • Mice
  • Nuclear Proteins / chemistry
  • Nuclear Proteins / metabolism*
  • Nuclear Receptor Coactivator 1
  • Nuclear Receptor Coactivator 2 / metabolism
  • Protein Binding
  • Protein Structure, Tertiary
  • Receptors, Estrogen / isolation & purification
  • Receptors, Estrogen / metabolism*
  • Transcription Factors / metabolism
  • Transcription, Genetic

Substances

  • GNL3L protein, mouse
  • Nuclear Proteins
  • Nuclear Receptor Coactivator 2
  • Receptors, Estrogen
  • Transcription Factors
  • estrogen receptor gamma
  • Histone Acetyltransferases
  • Ncoa1 protein, mouse
  • Nuclear Receptor Coactivator 1
  • GTP-Binding Proteins