Hematopoietic lineage cell specific protein 1 (HS1) is a functionally important signaling molecule in platelet activation

Blood. 2007 Oct 1;110(7):2449-56. doi: 10.1182/blood-2006-11-056069. Epub 2007 Jun 19.

Abstract

Collagen activates platelets through an intracellular signaling cascade downstream of glycoprotein VI (GPVI). We have investigated the contribution of hematopoietic lineage cell-specific protein 1 (HS1) downstream of GPVI in platelet activation. Stimulation of GPVI leads to tyrosine phosphorylation of HS1, which is blocked by Src-family kinase inhibitors. Coimmunoprecipitation experiments revealed that HS1 associates with Syk and phosphatidylinositol 3-kinases. HS1-null mice displayed increased bleeding times and increased time to occlusion in the FeCl(3) in vivo thrombosis model compared with their wild-type littermates. In addition, aggregation and secretion responses were diminished in HS1-null mouse platelets after stimulation of GPVI and protease-activated receptor 4 (PAR-4) agonists compared with wild-type littermate mouse platelets. Finally, Akt phosphorylation was diminished after GPVI or PAR-4 stimulation in platelets from HS1-null mice compared with their wild-type littermates. These results demonstrate that phosphorylation of the HS1 protein occurs downstream of GPVI stimulation and that HS1 plays a significant functional role in platelet activation downstream of GPVI and PARs.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Blood Platelets / metabolism*
  • Granulocyte Colony-Stimulating Factor / deficiency
  • Granulocyte Colony-Stimulating Factor / genetics
  • Granulocyte Colony-Stimulating Factor / metabolism*
  • Mice
  • Phosphatidylinositol 3-Kinases / metabolism
  • Phosphorylation / drug effects
  • Platelet Activation* / drug effects
  • Platelet Membrane Glycoproteins / metabolism
  • Protein Binding
  • Protein-Tyrosine Kinases / metabolism
  • Proto-Oncogene Proteins c-akt / agonists
  • Proto-Oncogene Proteins c-akt / metabolism
  • Purinergic P2 Receptor Antagonists
  • Receptors, Purinergic P2 / metabolism
  • Signal Transduction*

Substances

  • Platelet Membrane Glycoproteins
  • Purinergic P2 Receptor Antagonists
  • Receptors, Purinergic P2
  • hematopoietic lineage cell-specific protein 1, mouse
  • platelet membrane glycoprotein VI
  • Granulocyte Colony-Stimulating Factor
  • Phosphatidylinositol 3-Kinases
  • Protein-Tyrosine Kinases
  • Proto-Oncogene Proteins c-akt