Comparative modeling of the H4-H5-loop of the alpha2-isoform of Na+/K+-ATPase alpha-subunit in the E1 conformation

Physiol Res. 2007:56 Suppl 1:S143-S151. doi: 10.33549/physiolres.931313. Epub 2007 May 31.

Abstract

Restraint-based comparative modeling was used for calculation and visualization of the H4-H5-loop of Na+/K+-ATPase from mouse brain (Mus musculus, adult male brain, alpha2-isoform) between the amino acid residues Cys 336 and Arg 758 in the E1 conformation The structure consists of two well separated parts. The N-domain is formed by a seven-stranded antiparallel beta-sheet with two additional beta-strands and five alpha-helices sandwiching it, the P-domain is composed of a typical Rossman fold. The ATP-binding site was found on the N-domain to be identical in both alpha2- and alpha1-isoforms. The phosphorylation Asp 369 residue was found in the central part of the P-domain, located at the C-terminal end of the central beta-sheet. The distance between the alpha-carbon of Phe 475 at the ATP-binding site and the alpha-carbon of Asp 369 at the phosphorylation site is 3.22 nm. A hydrogen bond between the oxygen atom of Asp 369 and the nitrogen atom of Lys 690 was clearly detected and assumed to play a key role in maintaining the proper structure of the phosphorylaton site in E1 conformation.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Brain / enzymology*
  • Computer Graphics
  • Hydrogen Bonding
  • Imaging, Three-Dimensional
  • Isoenzymes / chemistry
  • Male
  • Mice
  • Models, Molecular*
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Conformation
  • Protein Structure, Tertiary
  • Reproducibility of Results
  • Sequence Alignment
  • Sequence Homology, Amino Acid
  • Sodium-Potassium-Exchanging ATPase / chemistry*
  • Sodium-Potassium-Exchanging ATPase / metabolism

Substances

  • Isoenzymes
  • Adenosine Triphosphate
  • Atp1a2 protein, mouse
  • Sodium-Potassium-Exchanging ATPase