Effects of 5-hydroxytryptamine on electrical responses of circular smooth muscle isolated from the guinea-pig gastric antrum

J Smooth Muscle Res. 2006 Dec;42(6):203-16. doi: 10.1540/jsmr.42.203.

Abstract

The effects of 5-hydroxytryptamine (5-HT) on electrical responses of the membrane were investigated in circular smooth muscle isolated from the guinea-pig stomach antrum. Small segment of circular muscle tissue produced a periodical generation of slow potentials at frequency of 0.1-2 cycles min(-1), during random generation of unitary potentials. Application of 5-HT (10(-7)-10(-5) M) hyperpolarized the membrane and either increased or decreased the frequency of slow potentials, both with associated increase in amplitude of slow potential. These effects of 5-HT were abolished by methysergide. N(omega)-nitro-L-arginine (L-NA) increased the frequency of spontaneously generated slow potentials and also increased the frequency of slow potentials generated during stimulation with 5-HT, suggesting an involvement of the increased production of nitric oxide (NO) by 5-HT. Atropine did not alter spontaneous and 5-HT-induced electrical responses. The hyperpolarization produced by 5-HT was associated with a decrease in input resistance and time constant of the membrane. The amplitude of the 5-HT-induced hyperpolarization was increased in low [K(+)](o) solution and decreased in high [K(+)](o) solution or in the presence of glybenclamide, suggesting that the hyperpolarization was produced by activation of ATP-sensitive K-channels. The increase in amplitude of slow potentials by 5-HT may be secondary due to hyperpolarization of the membrane. The inhibition by 5-HT of the frequency of slow potentials may be partly due to the increased release of NO, however the mechanism by which dual effects of 5-HT on the frequency of slow potentials remains unsolved.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Arrhythmia Agents / pharmacology
  • Atropine / pharmacology
  • Electrophysiology
  • Enzyme Inhibitors / pharmacology
  • Glyburide / pharmacology
  • Guinea Pigs
  • In Vitro Techniques
  • Male
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Methysergide / pharmacology
  • Muscle, Smooth / drug effects*
  • Muscle, Smooth / physiology*
  • Myenteric Plexus / drug effects
  • Myenteric Plexus / physiology
  • Nitroarginine / pharmacology
  • Parasympatholytics / pharmacology
  • Potassium / pharmacology
  • Pyloric Antrum / drug effects*
  • Pyloric Antrum / innervation
  • Pyloric Antrum / physiology
  • Serotonin / pharmacology*
  • Serotonin Agents / pharmacology*
  • Serotonin Antagonists / pharmacology

Substances

  • Anti-Arrhythmia Agents
  • Enzyme Inhibitors
  • Parasympatholytics
  • Serotonin Agents
  • Serotonin Antagonists
  • Nitroarginine
  • Serotonin
  • Atropine
  • Potassium
  • Glyburide
  • Methysergide