Nateglinide improves postprandial hyperglycemia and insulin secretion in renal transplant recipients

Clin Transplant. 2007 Mar-Apr;21(2):246-51. doi: 10.1111/j.1399-0012.2006.00634.x.

Abstract

Background: Postprandial hyperglycemia (PPHG) frequently occurs among renal transplant recipients (RTR). Reduced early insulin response (EIR) after a meal leads to impaired suppression of endogenous glucose production and subsequently PPHG, which is a risk factor for cardiovascular disease. Nateglinide is a rapid acting insulin secretagogue inducing an EIR after a meal. Our main objective was to investigate the safety and effect of nateglinide treatment on postprandial plasma glucose excursions and insulin secretion in RTR with PPHG.

Patients and methods: A total of 14 Caucasian RTR with new-onset diabetes mellitus (NODM; n = 6) or impaired glucose tolerance (IGT; n = 8) were included. The insulin response and glucose excursions were measured for 240 min after a standardized liquid meal at baseline and after two-wk treatment with nateglinide.

Results: Treatment with nateglinide was followed by a significant decrease in mean two-h plasma glucose from 10.5 mmol/L (3.1) to 7.6 mmol/L (2.1; p < 0.001) and a decline in total postprandial area under the curve (AUC) of glucose concentration (p < 0.001). Both estimated EIR and the late insulin response increased significantly (p = 0.008 and p = 0.003, respectively). No serious adverse event was observed during the study period.

Conclusions: Treating RTR with nateglinide for two-wk significantly improved PPHG, increased the insulin response following a standardized meal and was well tolerated.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Blood Glucose / drug effects*
  • Cyclohexanes / administration & dosage
  • Cyclohexanes / pharmacology*
  • Cyclohexanes / therapeutic use
  • Female
  • Humans
  • Hyperglycemia / prevention & control*
  • Hypoglycemic Agents / administration & dosage
  • Hypoglycemic Agents / pharmacology*
  • Hypoglycemic Agents / therapeutic use
  • Insulin / metabolism*
  • Insulin Secretion
  • Kidney Transplantation / physiology*
  • Male
  • Middle Aged
  • Nateglinide
  • Phenylalanine / administration & dosage
  • Phenylalanine / analogs & derivatives*
  • Phenylalanine / pharmacology
  • Phenylalanine / therapeutic use
  • Postprandial Period / drug effects*
  • Postprandial Period / physiology

Substances

  • Blood Glucose
  • Cyclohexanes
  • Hypoglycemic Agents
  • Insulin
  • Nateglinide
  • Phenylalanine