Microscopic intratumoral dosimetry of radiolabeled antibodies is a critical determinant of successful radioimmunotherapy in B-cell lymphoma

Cancer Res. 2007 Feb 1;67(3):1335-43. doi: 10.1158/0008-5472.CAN-06-2495.

Abstract

Radioimmunotherapy is a highly effective treatment for some hematologic malignancies; however, the underlying mechanisms of tumor clearance remain poorly understood. We have previously shown that both targeted radiation using (131)I-labeled anti-MHC class II (MHCII) monoclonal antibody (mAb) plus mAb signaling with unlabeled anti-idiotype are required for the long-term clearance of tumor in syngeneic murine lymphoma models. In this study, we have investigated how the microdistribution of the targeted radiation component of this combination affects the long-term clearance of lymphoma. (131)I-labeled mAb targeting CD45 and MHCII antigens was found to deliver similar doses of radiation to tumor-bearing organ using conventional dosimetry ( approximately 1.0 Gy per MBq when (131)I was labeled to 500 mug mAb and given i.v. per mouse), but when used as radiation vectors in combination therapy only, (131)I-anti-MHCII plus anti-idiotype produced long-term survival. The profound differences in therapy did not seem to be dependent on levels of (131)I-mAb tumor-binding or antibody-dependent cytotoxicity. Instead, the microscopic intratumoral dosimetry seemed to be critical with the (131)I-anti-MHCII, delivering more concentrated and therefore substantially higher radiation dose to tumor cells. When the administered activity of (131)I-anti-CD45 was increased, a radiation dose response was shown in the presence of anti-idiotype and long-term survival was seen. We believe that these new insights should influence the selection of new antigen targets and the design of dosimetric methods in radioimmunotherapy of lymphoma.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Monoclonal / administration & dosage
  • Antibodies, Monoclonal / immunology
  • Antibodies, Monoclonal / pharmacokinetics
  • Antibody-Dependent Cell Cytotoxicity
  • Histocompatibility Antigens Class II / immunology
  • Immunoconjugates / pharmacokinetics
  • Immunoconjugates / pharmacology
  • Iodine Radioisotopes / administration & dosage*
  • Leukocyte Common Antigens / immunology
  • Lymphoma, B-Cell / immunology
  • Lymphoma, B-Cell / radiotherapy*
  • Mice
  • Mice, Inbred BALB C
  • Radioimmunotherapy / methods*
  • Radiometry

Substances

  • Antibodies, Monoclonal
  • Histocompatibility Antigens Class II
  • Immunoconjugates
  • Iodine Radioisotopes
  • Leukocyte Common Antigens