Bone morphogenetic protein 7 (bmp-7) stimulates proteoglycan synthesis in human osteoarthritic chondrocytes in vitro

Biomed Pharmacother. 2006 Dec;60(10):639-43. doi: 10.1016/j.biopha.2006.09.001. Epub 2006 Oct 12.

Abstract

BMP-7 is a member of the TGF-beta superfamily which is supposed to be one of the most potent anabolic factors of chondrocytes. In this study we analysed the effect of BMP-7 on three dimensional cultured chondrocytes with and without serum. Cartilage samples from fourteen patients with osteoarthritis of the knee were harvested and chondrocytes were cultivated in alginate-beads with and without serum supplementation (10% FCS). BMP-7 was added in three different concentrations (200, 600 and 1000 ng/ml). After 4 and 21 days PG concentration was determined by a Blyscan-Assay. For gene expression analysis of aggrecan (AGG) quantitative Lightcycler-PCR was used to estimate the mRNA levels. Under serumfree culture conditions there was no stimulation after 4 days but there was a twofold increase of PG concentration after 21 days. Using BMP-7 together with serum supplemented medium we found comparable results, however not as pronounced. AGG expression was increased only after 4 days but not after 21 days. Beside a stimulatory effect under serumfree conditions we also found a stimulatory effect of BMP-7 in the presence of serum. This study pronounces that BMP-7 might be a suitable anabolic activator of osteoarthritic chondrocytes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Aggrecans / genetics
  • Aggrecans / metabolism
  • Alginates / chemistry
  • Bone Morphogenetic Protein 7
  • Bone Morphogenetic Proteins / pharmacology*
  • Cells, Cultured
  • Chondrocytes / drug effects*
  • Chondrocytes / metabolism
  • Chondrocytes / pathology
  • Culture Media, Serum-Free / pharmacology
  • Dose-Response Relationship, Drug
  • Gene Expression / drug effects
  • Glucuronic Acid / chemistry
  • Hexuronic Acids / chemistry
  • Humans
  • Microspheres
  • Middle Aged
  • Osteoarthritis, Knee / pathology
  • Proteoglycans / biosynthesis*
  • Proteoglycans / genetics
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Reverse Transcriptase Polymerase Chain Reaction
  • Time Factors
  • Transforming Growth Factor beta / pharmacology*

Substances

  • Aggrecans
  • Alginates
  • BMP7 protein, human
  • Bone Morphogenetic Protein 7
  • Bone Morphogenetic Proteins
  • Culture Media, Serum-Free
  • Hexuronic Acids
  • Proteoglycans
  • RNA, Messenger
  • Transforming Growth Factor beta
  • Glucuronic Acid