Antiaggressive effects of MPEP, a selective antagonist of mGlu5 receptors, in agonistic interactions between male mice

Eur J Pharmacol. 2006 Dec 3;551(1-3):67-70. doi: 10.1016/j.ejphar.2006.08.055. Epub 2006 Sep 8.

Abstract

mGlu5 receptors are highly concentrated in limbic brain structures involved in motivational and emotional behaviours. This study describes the effects of 2-methyl-6-(phenylethylnyl)pyridine (MPEP; 5, 10, 15, 20 and 25 mg/kg, ip), a selective antagonist of the mGlu5 receptors, on agonistic behaviour elicited by isolation in male mice. Individually housed mice were exposed to anosmic opponents in a neutral area 30 min after drug administration. Besides other behaviours, the aggressive (threat and attack) and exploratory behaviours were evaluated during 10 min using an ethologically based analysis. MPEP produced a behavioural profile characterized by a notable decrement of offensive behaviours, accompanied by a significant increase of exploratory behaviours (nonsocial exploration and social investigation). These findings suggest a role for mGlu5 receptors in aggression modulation.

MeSH terms

  • Aggression / drug effects
  • Agonistic Behavior / drug effects*
  • Animals
  • Behavior, Animal / drug effects*
  • Brain / drug effects*
  • Brain / metabolism
  • Dose-Response Relationship, Drug
  • Excitatory Amino Acid Antagonists / pharmacology*
  • Exploratory Behavior / drug effects
  • Male
  • Mice
  • Pyridines / pharmacology*
  • Receptor, Metabotropic Glutamate 5
  • Receptors, Metabotropic Glutamate / antagonists & inhibitors*
  • Receptors, Metabotropic Glutamate / metabolism

Substances

  • Excitatory Amino Acid Antagonists
  • Pyridines
  • Receptor, Metabotropic Glutamate 5
  • Receptors, Metabotropic Glutamate
  • 6-methyl-2-(phenylethynyl)pyridine