Effect of fluticasone propionate/salmeterol on lung hyperinflation and exercise endurance in COPD

Chest. 2006 Sep;130(3):647-56. doi: 10.1378/chest.130.3.647.

Abstract

Study objective: To examine the effect of fluticasone propionate, 250 microg/salmeterol, 50 microg combination (FSC 250/50) twice daily on lung hyperinflation and associated measures of exercise performance in patients with COPD.

Design: This was a randomized, double-blind, parallel-group study.

Patients: Eligible patients were > or = 40 years old with a diagnosis of COPD, prealbuterol FEV(1) < 70% of predicted, FEV1/FVC ratio > or = 0.70, and functional residual capacity (FRC) > or = 120% of predicted normal.

Interventions: Patients were randomized to FSC 250/50; salmeterol, 50 microg; or placebo twice daily for 8 weeks. Predose and postdose spirometry, plethysmography, and constant-load cycle cardiopulmonary exercise test evaluations were compared. The primary comparison was FSC 250/50 with placebo. The salmeterol group was included for exploratory comparisons with FSC 250/50.

Results: A total of 185 patients (mean baseline FEV1 of 41% predicted) were enrolled. At rest, FSC 250/50 significantly reduced postdose FRC and increased inspiratory capacity (IC) compared with placebo (differences of - 0.35 +/- 0.12 L and 0.33 +/- 0.06 L [mean +/- SE], respectively, at week 8; p > or = 0.003) and increased exercise endurance time (difference, 132 +/- 45 s; p = 0.004). At a standardized time during exercise (isotime), FSC 250/50 increased postdose IC by 0.20 +/- 0.05 L over placebo with associated improvements in tidal volume and minute ventilation (p < 0.05 vs placebo at week 8). Improvement in exercise time was significantly correlated with the increase in IC (r = 0.45, p < 0.001) but not FEV1 (r = 0.23, p = 0.08). Predose comparisons of FSC 250/50 with salmeterol and placebo favored FSC 250/50.

Conclusion: We conclude that FSC 250/50 decreases lung hyperinflation at rest and during exercise with an associated increase in exercise endurance time when compared with placebo.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic beta-Agonists / adverse effects
  • Adrenergic beta-Agonists / pharmacology
  • Adrenergic beta-Agonists / therapeutic use
  • Aged
  • Albuterol / adverse effects
  • Albuterol / analogs & derivatives*
  • Albuterol / pharmacology
  • Albuterol / therapeutic use
  • Androstadienes / adverse effects
  • Androstadienes / pharmacology*
  • Androstadienes / therapeutic use*
  • Bronchodilator Agents / adverse effects
  • Bronchodilator Agents / pharmacology*
  • Bronchodilator Agents / therapeutic use*
  • Dose-Response Relationship, Drug
  • Double-Blind Method
  • Drug Combinations
  • Dyspnea / physiopathology
  • Female
  • Fluticasone-Salmeterol Drug Combination
  • Humans
  • Lung / drug effects*
  • Lung / pathology
  • Lung / physiopathology
  • Lung Volume Measurements
  • Male
  • Middle Aged
  • Physical Endurance / drug effects*
  • Physical Endurance / physiology
  • Pulmonary Disease, Chronic Obstructive / drug therapy*
  • Pulmonary Disease, Chronic Obstructive / pathology
  • Pulmonary Disease, Chronic Obstructive / physiopathology
  • Pulmonary Ventilation / drug effects
  • Pulmonary Ventilation / physiology
  • Respiratory Function Tests
  • Respiratory Mechanics / drug effects
  • Respiratory Mechanics / physiology
  • Salmeterol Xinafoate
  • Tidal Volume / drug effects
  • Tidal Volume / physiology
  • Time Factors

Substances

  • Adrenergic beta-Agonists
  • Androstadienes
  • Bronchodilator Agents
  • Drug Combinations
  • Fluticasone-Salmeterol Drug Combination
  • Salmeterol Xinafoate
  • Albuterol