Peptide bond formation does not involve acid-base catalysis by ribosomal residues

Nat Struct Mol Biol. 2006 May;13(5):423-8. doi: 10.1038/nsmb1091. Epub 2006 Apr 30.

Abstract

Ribosomes catalyze the formation of peptide bonds between aminoacyl esters of transfer RNAs within a catalytic center composed of ribosomal RNA only. Here we show that the reaction of P-site formylmethionine (fMet)-tRNA(fMet) with a modified A-site tRNA substrate, Phelac-tRNA(Phe), in which the nucleophilic amino group is replaced with a hydroxyl group, does not show the pH dependence observed with small substrate analogs such as puromycin and hydroxypuromycin. This indicates that acid-base catalysis by ribosomal residues is not important in the reaction with the full-size substrate. Rather, the ribosome catalyzes peptide bond formation by positioning the tRNAs, or their 3' termini, through interactions with rRNA that induce and/or stabilize a pH-insensitive conformation of the active site and provide a preorganized environment facilitating the reaction. The rate of peptide bond formation with unmodified Phe-tRNA(Phe) is estimated to be >300 s(-1).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acids / chemistry
  • Alkalies / chemistry
  • Catalysis
  • Hydrogen-Ion Concentration
  • Kinetics
  • Peptides / chemistry*
  • Peptides / metabolism*
  • Peptidyl Transferases / metabolism
  • Protein Biosynthesis*
  • RNA, Transfer / metabolism
  • Ribosomes / genetics*
  • Ribosomes / metabolism*
  • Substrate Specificity
  • Transfer RNA Aminoacylation

Substances

  • Acids
  • Alkalies
  • Peptides
  • RNA, Transfer
  • Peptidyl Transferases