Self-assembly of HEK cell-secreted ApoE particles resembles ApoE enrichment of lipoproteins as a ligand for the LDL receptor-related protein

Biochemistry. 2006 Jan 17;45(2):381-90. doi: 10.1021/bi051765s.

Abstract

Recent studies have shown that the lipidation and assembly state of apolipoprotein E (apoE) determine receptor recognition and amyloid-beta peptide (Abeta) binding. We previously demonstrated that apoE secreted by HEK cells stably expressing apoE3 or apoE4 (HEK-apoE) binds Abeta and inhibits Abeta-induced neurotoxicity by an isoform-specific process that requires apoE receptors. Here we characterized the structure of HEK-apoE assemblies and determined their receptor binding specificity. By chromatography, HEK-apoE elutes in high molecular mass fractions and is the size of plasma HDL, consistent with a multiprotein assembly. No lipid was associated with these apoE assemblies. Several methods for analyzing receptor binding indicate that HEK-apoE is a ligand for low-density lipoprotein (LDL) receptor-related protein (LRP) but not the LDL receptor. This suggests that self-assembly of apoE may induce a functional conformation necessary for binding to LRP. Our results indicate that, in addition to lipid content, the assembly state of apoE influences Abeta binding and receptor recognition.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apolipoprotein E3
  • Apolipoprotein E4
  • Apolipoproteins E / chemistry*
  • Apolipoproteins E / metabolism*
  • Apolipoproteins E / ultrastructure
  • Cell Line
  • Chromatography, Gel
  • Fibroblasts / metabolism
  • Humans
  • Iodine Radioisotopes
  • Ligands
  • Low Density Lipoprotein Receptor-Related Protein-1 / chemistry
  • Low Density Lipoprotein Receptor-Related Protein-1 / metabolism*
  • Mice
  • Protein Binding
  • Receptors, LDL / metabolism
  • Ultracentrifugation

Substances

  • Apolipoprotein E3
  • Apolipoprotein E4
  • Apolipoproteins E
  • Iodine Radioisotopes
  • Ligands
  • Low Density Lipoprotein Receptor-Related Protein-1
  • Receptors, LDL