Two different Ca2+ ion binding sites in factor VIIa and in des(1-38) factor VIIa

FEBS Lett. 1992 Jul 20;306(2-3):265-8. doi: 10.1016/0014-5793(92)81014-d.

Abstract

The Ca2+ ion binding of factor VIIa and the derivative lacking the gamma-carboxyglutamic acid domain, des(1-38) factor VIIa, was investigated using intrinsic protein fluorescence and Tb3+ ion phosphorescence methods. Binding of Ca2+ ions giving rise to a decrease in the intrinsic protein fluorescence (approximately 50% at saturating conditions) is seen with both proteins. Each of the saturation curves is in accordance with the formation of a 1:1 complex of factor VIIa-Ca2+ (KD approximately 30 microM) and des(1-38) factor VIIa-Ca2+ (KD approximately 40 microM)). Yet another Ca2+ ion binding site reveals itself in each protein in Tb3+ ion phosphorescence experiments. Ca2+ ion competition studies have showed 1:1 complexes (KD's approximately 2 mM). The results are interpreted in terms of two different Ca2+ ion binding sites, one in the EGF-1 domain and one in the Gly-209-Gln-221 loop of the serine proteinase part.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding Sites
  • Calcium / metabolism*
  • Cell Line
  • Cricetinae
  • Factor VIIa / chemistry
  • Factor VIIa / metabolism*
  • Humans
  • Peptide Fragments / chemistry
  • Peptide Fragments / metabolism*
  • Spectrometry, Fluorescence
  • Terbium / metabolism

Substances

  • Peptide Fragments
  • des(1-38) factor VIIa
  • Terbium
  • Factor VIIa
  • Calcium