[Adefovir dipivoxil in treatment of decompensated liver cirrhosis patients with YMDD mutation]

Zhejiang Da Xue Xue Bao Yi Xue Ban. 2005 Sep;34(5):470-2. doi: 10.3785/j.issn.1008-9292.2005.05.018.
[Article in Chinese]

Abstract

Objective: To evaluate the efficacy and safety of adefovir dipivoxil in treatment of decompensated liver cirrhosis patients with YMDD motif mutation during lamivudine therapy.

Methods: The disease relapsed in 14 hepatitis B patients with decompensated liver cirrhosis during lamivudine treatment due to the YMDD motif mutation. All 14 patients had positive HVBDNA and active hepatitis, and were evaluated as Child-Pugh Score C (CPS-C). The patients were treated with lamivudine 50 mg/d and adefovir dipivoxil 10 mg/d for 6 months.

Results: One patient signed off due to non-hypoxemic hyperlactacidemia; other 13 patients showed decreased serum HBVDNA. All patients had serum HBVDNA < or =10(5) copies/ml and 7 patients had HBVDNA < or =10(4) copies/ml. Six patients regained normal serum ALT level and Child-Pugh scores decreased in all patients.

Conclusion: Adefovir dipivoxil has satisfied efficacy and safety in treatment of decompensated liver cirrhosis patients with YMDD motif mutation during lamivudine treatment.

Publication types

  • English Abstract

MeSH terms

  • Adenine / adverse effects
  • Adenine / analogs & derivatives*
  • Adenine / therapeutic use
  • Adult
  • Aged
  • Amino Acid Motifs / genetics
  • Antiviral Agents / therapeutic use
  • DNA-Directed DNA Polymerase / genetics
  • Female
  • Hepatic Encephalopathy / drug therapy*
  • Hepatic Encephalopathy / genetics
  • Hepatic Encephalopathy / virology
  • Hepatitis B virus / genetics
  • Hepatitis B, Chronic / complications
  • Hepatitis B, Chronic / drug therapy
  • Humans
  • Lamivudine / therapeutic use
  • Liver Cirrhosis / drug therapy*
  • Liver Cirrhosis / genetics*
  • Liver Cirrhosis / virology
  • Male
  • Middle Aged
  • Mutation*
  • Organophosphonates / adverse effects
  • Organophosphonates / therapeutic use*
  • Protein Structure, Tertiary / genetics
  • Recurrence
  • Reverse Transcription / genetics

Substances

  • Antiviral Agents
  • Organophosphonates
  • Lamivudine
  • DNA-Directed DNA Polymerase
  • Adenine
  • adefovir dipivoxil