Induction of unstable and stable chromosomal aberrations by 99mTc: in-vitro and in-vivo studies

Nucl Med Commun. 2005 Oct;26(10):913-8. doi: 10.1097/00006231-200510000-00010.

Abstract

Background: Biological dosimetry, which determines the dose of acquired radiation by measuring radiation-induced variation of biological parameters, can help assess radiation damage in an individual. Evaluation of radiation exposure requires setting up reference curves for each type of radiation.

Aim: To evaluate the potential induction of chromosome aberrations by a clinical diagnostic dose of 99mTc.

Methods: Dicentrics, rings, excess fragments, complete reciprocal translocations and incomplete reciprocal translocations were scored in peripheral blood lymphocytes from patients exposed to a 99mTc bone scintigraphy. A specific relationship between the radiation dose delivered by 99mTc and the frequency of stable and unstable chromosomal aberrations was established in vitro to estimate whole-body dose. Chromosome analysis using fluorescence plus Giemsa and fluorescence in-situ hybridization was undertaken on six patients before and after a 99mTc bone scintigraphy. Dicentrics, rings, excess fragments, and translocations were scored in blood lymphocytes after in vitro 99mTc external irradiation in order to construct dose calibration curves.

Results: Analysis of the in-vitro data shows that the number of both unstable and stable aberrations has a quadratic linear relationship to the dose. Our in-vivo irradiation studies showed that activities of 99mTc-hexamethylene diphosphonate (99mTc-HDP) used for bone investigations do not induce any additional unstable chromosome aberrations and translocations. The frequencies obtained did not differ significantly from background values.

Conclusions: 99mTc can produce unstable and stable chromosomal aberrations in vitro. 99mTc-HDP administration does not induce supplementary chromosomal aberrations. The dose-response curves will allow a more accurate evaluation of the risk related to in-vivo administration of 99mTc labelled radiopharmaceuticals, and they can be used to assess the safe upper limit of injected activity in humans.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Chromosome Aberrations / radiation effects*
  • Chromosomes, Human / genetics*
  • Chromosomes, Human / radiation effects*
  • Dose-Response Relationship, Radiation
  • Humans
  • Radiation Dosage
  • Radiation Injuries / etiology*
  • Radiation Injuries / genetics*
  • Radiopharmaceuticals / adverse effects
  • Risk Assessment / methods*
  • Risk Factors
  • Technetium / adverse effects*

Substances

  • Radiopharmaceuticals
  • Technetium