Evidence for a functional interaction of the angiotensin-(1-7) receptor Mas with AT1 and AT2 receptors in the mouse heart

Hypertension. 2005 Oct;46(4):937-42. doi: 10.1161/01.HYP.0000175813.04375.8a. Epub 2005 Sep 12.

Abstract

The aim of this study was to evaluate the angiotensin (Ang)-(1-7) effects in isolated mouse hearts. The hearts of male C57BL/6J and knockout mice for the Ang-(1-7) receptor Mas were perfused by the Langendorff method. After a basal period, the hearts were perfused for 20 minutes with Krebs-Ringer solution (KRS) alone (control) or KRS containing Ang-(1-7) (0.22 pmol/L), the Mas antagonist A-779 (115 nmol/L), the angiotensin type 1 receptor antagonist losartan (2.2 micromol/L), or the angiotensin type 2 receptor antagonist PD123319 (130 nmol/L). To evaluate the involvement of Ang receptors, prostaglandins, and nitric oxide in the Ang-(1-7) effects, the hearts were perfused for 20 to 30 minutes with KRS containing either A-779, losartan, PD123319, indomethacin, or NG-nitro-L-arginine methyl ester (L-NAME) alone or in association with subsequent Ang-(1-7) perfusion. In addition, hearts from Mas-knockout mice were perfused for 20 minutes with KRS containing Ang-(1-7) (0.22 pmol/L) and losartan. Ang-(1-7) alone did not change the perfusion pressure. Strikingly, in the presence of losartan, 0.22 pmol/L Ang-(1-7) induced a significant decrease in perfusion pressure, which was blocked by A-779, indomethacin, and L-NAME. Furthermore, this effect was not observed in Mas-knockout mice. In contrast, in the presence of PD123319, Ang-(1-7) produced a significant increase in perfusion pressure. This change was not modified by the addition of A-779. Losartan reduced but did not abolish this effect. Our results suggest that Ang-(1-7) produces complex vascular effects in isolated, perfused mouse hearts involving interaction of its receptor with angiotensin type 1- and type 2-related mechanisms, leading to the release of prostaglandins and nitric oxide.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiotensin I / pharmacology
  • Angiotensin II / analogs & derivatives
  • Angiotensin II / pharmacology
  • Angiotensin II Type 1 Receptor Blockers / pharmacology
  • Animals
  • Drug Synergism
  • Enzyme Inhibitors / pharmacology
  • Imidazoles / pharmacology
  • In Vitro Techniques
  • Indomethacin / pharmacology
  • Losartan / pharmacology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Myocardium / metabolism*
  • NG-Nitroarginine Methyl Ester / pharmacology
  • Peptide Fragments / pharmacology
  • Perfusion
  • Pressure
  • Proto-Oncogene Mas
  • Proto-Oncogene Proteins / physiology*
  • Pyridines / pharmacology
  • Receptor, Angiotensin, Type 1 / drug effects*
  • Receptor, Angiotensin, Type 2 / drug effects*
  • Receptors, G-Protein-Coupled / physiology*
  • Vasoconstrictor Agents / pharmacology

Substances

  • 7-Ala-angiotensin (1-7)
  • Angiotensin II Type 1 Receptor Blockers
  • Enzyme Inhibitors
  • Imidazoles
  • Peptide Fragments
  • Proto-Oncogene Mas
  • Proto-Oncogene Proteins
  • Pyridines
  • Receptor, Angiotensin, Type 1
  • Receptor, Angiotensin, Type 2
  • Receptors, G-Protein-Coupled
  • Vasoconstrictor Agents
  • Angiotensin II
  • PD 123319
  • Angiotensin I
  • angiotensin I (1-7)
  • Losartan
  • NG-Nitroarginine Methyl Ester
  • Indomethacin