Studies on absorption and hydrolysis of ethyl alpha-D-glucoside in rat intestine

J Agric Food Chem. 2005 Sep 7;53(18):7257-61. doi: 10.1021/jf0508753.

Abstract

Ethyl alpha-D-glucoside (alpha-EG) is normally contained in Sake, which has been taken by Japanese people since ancient times. In this study, the intestinal absorption of alpha-EG was investigated using rat everted intestinal sac. Furthermore, the alpha-EG hydrolytic activity in rat intestine was compared with disaccharides hydrolytic activities, and the effects of alpha-EG on disaccharides hydrolysis were examined using crude enzyme preparation from rat intestinal acetone powder. Glucose liberated from alpha-EG was detected in a serosal solution of everted rat intestinal sac, but it was only less than 4% of absorbed intact alpha-EG. alpha-EG absorption into small intestinal tissue was reduced by elimination of sodium ion from the mucosal solution or under the presence of phlorizin. The hydrolytic activity for alpha-EG was detected in crude enzyme preparation from rat intestinal acetone powder, but it showed a low value as compared to those for disaccharides. alpha-EG showed mixed type inhibition for maltose and sucrose hydrolysis, but inhibitory concentrations of alpha-EG required for 50% inhibition for the maltose and sucrose hydrolysis were higher than those of arabinose and acarbose. In conclusion, a small amount of alpha-EG was hydrolyzed and most of it was absorbed via SGLT1 as an intact form in the rat small intestine, and the inhibitory effect of alpha-EG on disaccharides hydrolysis was weak.

MeSH terms

  • Animals
  • Disaccharides / metabolism
  • Glucose / metabolism
  • Glucosides / metabolism
  • Glucosides / pharmacokinetics*
  • Glucosides / pharmacology
  • Hydrolysis / drug effects
  • Intestinal Absorption*
  • Intestines / enzymology*
  • Kinetics
  • Rats
  • Rats, Wistar

Substances

  • Disaccharides
  • Glucosides
  • ethyl glucoside
  • Glucose